Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50013764
TargetProtein tyrosine phosphatase type IVA 3(Human)
Shanxi University

Curated by ChEMBL
LigandPNGBDBM396097(US10308663, JMS-631-053 | US12227515, Compound JMS...)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human His6-tagged PRL-3 expressed in Escherichia coli using DiFMUP as substrate incubated for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein tyrosine phosphatase type IVA 1(Human)
Shanxi University

Curated by ChEMBL
LigandPNGBDBM50059084(CHEMBL3393171 | US10308663, Thienopyridone (5))
Affinity DataIC50: 130nMAssay Description:Inhibition of full-length human brain His6-tagged PRL-1 expressed in Escherichia coli using TAMRA-Thr-Ala-Asp-Ile-Tyr(PO3H2)-Glu-NH2 peptide as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein tyrosine phosphatase type IVA 2(Human)
Shanxi University

Curated by ChEMBL
LigandPNGBDBM50059084(CHEMBL3393171 | US10308663, Thienopyridone (5))
Affinity DataIC50: 130nMAssay Description:Inhibition of human His6-tagged PRL-2 expressed in Escherichia coli using TAMRA-Thr-Ala-Asp-Ile-Tyr(PO3H2)-Glu-NH2 peptide as substrate by IMAP-FP as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein tyrosine phosphatase type IVA 3(Human)
Shanxi University

Curated by ChEMBL
LigandPNGBDBM50059084(CHEMBL3393171 | US10308663, Thienopyridone (5))
Affinity DataIC50: 460nMAssay Description:Inhibition of full-length human heart His6-tagged PRL-3 expressed in Escherichia coli using DiFMUP as substrate incubated for 35 mins by fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein tyrosine phosphatase type IVA 3(Human)
Shanxi University

Curated by ChEMBL
LigandPNGBDBM50569365(CHEMBL4867742)
Affinity DataIC50: 1.52E+4nMAssay Description:Inhibition of PRL-3 (unknown origin) using DiFMUP as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein tyrosine phosphatase type IVA 3(Human)
Shanxi University

Curated by ChEMBL
LigandPNGBDBM50569366(CHEMBL4858539)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of PRL-3 (unknown origin) using DiFMUP as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein tyrosine phosphatase type IVA 3(Human)
Shanxi University

Curated by ChEMBL
LigandPNGBDBM50323199(5,7-dihydroxy-8-(5-(5-hydroxy-7-methoxy-4-oxo-4H-c...)
Affinity DataIC50: 2.58E+4nMAssay Description:Inhibition of human brain PRL-3 (1 to 168 residues) expressed in Escherichia coli BL21(DE3) cells using DiFMUP as substrate incubated for 1 hr by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein tyrosine phosphatase type IVA 3(Human)
Shanxi University

Curated by ChEMBL
LigandPNGBDBM50569362(CHEMBL1699070)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of PRL-3 (unknown origin) using DiFMUP as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein tyrosine phosphatase type IVA 3(Human)
Shanxi University

Curated by ChEMBL
LigandPNGBDBM50569367(CHEMBL4850661)
Affinity DataIC50: 2.67E+4nMAssay Description:Inhibition of PRL-3 (unknown origin) using DiFMUP as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein tyrosine phosphatase type IVA 3(Human)
Shanxi University

Curated by ChEMBL
LigandPNGBDBM50323206(sciadopitisin | sciadopitysin | CHEMBL208908)
Affinity DataIC50: 4.62E+4nMAssay Description:Inhibition of human brain PRL-3 (1 to 168 residues) expressed in Escherichia coli BL21(DE3) cells using DiFMUP as substrate incubated for 1 hr by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein tyrosine phosphatase type IVA 3(Human)
Shanxi University

Curated by ChEMBL
LigandPNGBDBM50569368(CHEMBL4876462)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of PRL-3 (unknown origin) using DiFMUP as substrate incubated for 5 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein tyrosine phosphatase type IVA 3(Human)
Shanxi University

Curated by ChEMBL
LigandPNGBDBM50569363(CHEMBL4878327)
Affinity DataIC50: 8.87E+4nMAssay Description:Inhibition of PRL-3 (unknown origin) using DiFMUP as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProtein tyrosine phosphatase type IVA 3(Human)
Shanxi University

Curated by ChEMBL
LigandPNGBDBM50569364(CHEMBL4848603)
Affinity DataIC50: 9.84E+4nMAssay Description:Inhibition of PRL-3 (unknown origin) using DiFMUP as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed