Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50013475
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566369(CHEMBL4859651)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566366(CHEMBL4854804)
Affinity DataEC50:  0.25nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566365(CHEMBL4848974)
Affinity DataEC50:  0.380nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566372(CHEMBL4859407)
Affinity DataEC50:  0.410nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566373(CHEMBL4847662)
Affinity DataEC50:  0.417nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566374(CHEMBL4872298)
Affinity DataEC50:  0.729nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566368(CHEMBL4857550)
Affinity DataEC50:  0.730nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566357(CHEMBL4874972)
Affinity DataEC50:  2nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566362(CHEMBL4869870)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566359(CHEMBL4855306)
Affinity DataEC50:  4.80nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566358(Mk-8666)
Affinity DataEC50:  5.60nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566355(CHEMBL4868224)
Affinity DataEC50:  14nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566367(CHEMBL4858086)
Affinity DataEC50:  16nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566360(CHEMBL4866406)
Affinity DataEC50:  21nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566370(CHEMBL4877893)
Affinity DataEC50: >25nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566371(CHEMBL4868676)
Affinity DataEC50: >25nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566375(CHEMBL4865460)
Affinity DataEC50: >25nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566376(CHEMBL4850966)
Affinity DataEC50: >25nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566361(CHEMBL4852222)
Affinity DataEC50: >25nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566363(CHEMBL4866568)
Affinity DataEC50: >25nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566364(CHEMBL4852865)
Affinity DataEC50: >25nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM22496(CHEMBL207881 | 3-(4-{[(3-phenoxyphenyl)methyl]amin...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50392861(CHEMBL2152070)
Affinity DataEC50:  160nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566356(CHEMBL4846948)
Affinity DataEC50:  233nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566369(CHEMBL4859651)
Affinity DataEC50:  521nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/CRE (Gs) assessed as firefly luciferase activity at 10 uM incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566369(CHEMBL4859651)
Affinity DataEC50:  681nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells assessed as increase in cAMP level incubated for 30 mins by cAMP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566373(CHEMBL4847662)
Affinity DataEC50:  7.53E+3nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells assessed as increase in cAMP level incubated for 30 mins by cAMP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566373(CHEMBL4847662)
Affinity DataEC50:  1.29E+4nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/CRE (Gs) assessed as firefly luciferase activity at 10 uM incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566373(CHEMBL4847662)
Affinity DataEC50:  1.48E+4nMAssay Description:Agonist activity at FFAR4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 2(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566373(CHEMBL4847662)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at FFAR2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 3(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566369(CHEMBL4859651)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at FFAR3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 3(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566373(CHEMBL4847662)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at FFAR3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566369(CHEMBL4859651)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at FFAR4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetFree fatty acid receptor 2(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566369(CHEMBL4859651)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at FFAR2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566366(CHEMBL4854804)
Affinity DataEC50:  2.78E+4nMAssay Description:Agonist activity at human PPARgamma expressed in CHO cells assessed as increase in receptor transcriptional activity incubated for 24 hrs by dual luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50566369(CHEMBL4859651)
Affinity DataEC50:  5.69E+4nMAssay Description:Agonist activity at human PPARgamma expressed in CHO cells assessed as increase in receptor transcriptional activity incubated for 24 hrs by dual luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed