Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50013212
TargetInterleukin-1 receptor-associated kinase 4(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50563725(CHEMBL4761018 | US12304916, Example 79)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of IRAK4 (unknown origin) using IPTSPITTTYFFFKKK peptide as substrate in presence of ATP measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50563729(CHEMBL4749904 | US12304916, Example 21)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of IRAK4 (unknown origin) using IPTSPITTTYFFFKKK peptide as substrate in presence of ATP measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50563726(CHEMBL4754408 | US12304916, Example 45)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of IRAK4 (unknown origin) using IPTSPITTTYFFFKKK peptide as substrate in presence of ATP measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50563727(CHEMBL4762550 | US12304916, Example 59)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of IRAK4 (unknown origin) using IPTSPITTTYFFFKKK peptide as substrate in presence of ATP measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50563728(CHEMBL4756721 | US12304916, Example 23)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of IRAK4 (unknown origin) using IPTSPITTTYFFFKKK peptide as substrate in presence of ATP measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50563724(CHEMBL4789541 | US12304916, Example 80)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of IRAK4 (unknown origin) using IPTSPITTTYFFFKKK peptide as substrate in presence of ATP measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed