Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50014421
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50069799(CHEMBL3407579 | US9187441, 7M)
Affinity DataKi:  400nMAssay Description:Displacement of fluorescent F4 peptide from MDM2 (1 to 125 residues) (unknown origin) expressed in Escherichia coli by fluorescence polarization assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50069799(CHEMBL3407579 | US9187441, 7M)
Affinity DataKi:  800nMAssay Description:Displacement of 5-FAM labeled PMDM6-F from GST-tagged human recombinant MDM2 (1 to 118 residues) expressed in Escherichia coli incubated for 0.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50576033(CHEMBL4847555)
Affinity DataKi:  9.20E+3nMAssay Description:Displacement of 5-FAM labeled PMDM6-F from GST-tagged human recombinant MDM2 (1 to 118 residues) expressed in Escherichia coli incubated for 0.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed