Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50013913
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570832(CHEMBL4848594)
Affinity DataEC50:  12nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570834(CHEMBL4877644 | US11918568, Example 9)
Affinity DataEC50:  22nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570846(CHEMBL4847819)
Affinity DataIC50: 32nMAssay Description:Inhibition of human NAMPT assessed as decrease in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570831(CHEMBL4846468 | US11918568, Example 26)
Affinity DataEC50:  40nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570836(CHEMBL4860172)
Affinity DataEC50:  70nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570833(CHEMBL4861097 | US11918568, Example 8)
Affinity DataEC50:  83nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570844(CHEMBL4877360)
Affinity DataEC50:  83nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570841(CHEMBL4872409)
Affinity DataEC50:  120nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570835(CHEMBL4858166 | US11918568, Example 10)
Affinity DataEC50:  140nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570842(CHEMBL4868811 | US11918568, Example 13)
Affinity DataEC50:  180nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570843(CHEMBL4861428)
Affinity DataEC50:  190nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570829(CHEMBL4872450)
Affinity DataEC50:  220nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570837(CHEMBL4873608)
Affinity DataEC50:  350nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570828(CHEMBL4864574)
Affinity DataEC50:  480nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570830(CHEMBL4872111 | US11918568, Example 32)
Affinity DataEC50:  510nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570845(CHEMBL4877613)
Affinity DataEC50:  530nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570840(CHEMBL4845888)
Affinity DataEC50:  2.40E+3nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50569506(CHEMBL1520901 | US11452717, Compound TableB-2.28)
Affinity DataEC50:  3.30E+3nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570839(CHEMBL4879270)
Affinity DataEC50:  5.80E+3nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570838(CHEMBL4860234)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of human NAMPT assessed as increase in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed