Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50013916
TargetAminopeptidase N(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570849(CHEMBL4854733)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570849(CHEMBL4854733)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570850(CHEMBL4877339)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570850(CHEMBL4877339)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570851(CHEMBL4853049)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570851(CHEMBL4853049)
Affinity DataIC50: 8.70nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human ERAP2 using R-AMC as substrate incubated for 5 to 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEndoplasmic reticulum aminopeptidase 1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 33nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate incubated for 5 to 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEndoplasmic reticulum aminopeptidase 1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570849(CHEMBL4854733)
Affinity DataIC50: 140nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570849(CHEMBL4854733)
Affinity DataIC50: 141nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 186nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEndoplasmic reticulum aminopeptidase 1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 190nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAminopeptidase N(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570847(CHEMBL4863168)
Affinity DataIC50: 224nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570847(CHEMBL4863168)
Affinity DataIC50: 230nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570851(CHEMBL4853049)
Affinity DataIC50: 324nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570851(CHEMBL4853049)
Affinity DataIC50: 330nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570850(CHEMBL4877339)
Affinity DataIC50: 410nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570850(CHEMBL4877339)
Affinity DataIC50: 417nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570849(CHEMBL4854733)
Affinity DataIC50: 891nMAssay Description:Inhibition of ERAP2 (unknown origin) using R-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570849(CHEMBL4854733)
Affinity DataIC50: 900nMAssay Description:Inhibition of ERAP2 (unknown origin) using R-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570851(CHEMBL4853049)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of ERAP2 (unknown origin) using R-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570851(CHEMBL4853049)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of ERAP2 (unknown origin) using R-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570850(CHEMBL4877339)
Affinity DataIC50: 2.34E+3nMAssay Description:Inhibition of ERAP2 (unknown origin) using R-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570850(CHEMBL4877339)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of ERAP2 (unknown origin) using R-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 2.95E+3nMAssay Description:Inhibition of ERAP2 (unknown origin) using R-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEndoplasmic reticulum aminopeptidase 2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of ERAP2 (unknown origin) using R-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAminopeptidase N(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570848(CHEMBL4872604)
Affinity DataIC50: 3.39E+3nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570848(CHEMBL4872604)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570847(CHEMBL4863168)
Affinity DataIC50: 1.74E+4nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570847(CHEMBL4863168)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570848(CHEMBL4872604)
Affinity DataIC50: 7.70E+4nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570848(CHEMBL4872604)
Affinity DataIC50: 7.76E+4nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570847(CHEMBL4863168)
Affinity DataIC50: 9.77E+4nMAssay Description:Inhibition of ERAP2 (unknown origin) using R-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570847(CHEMBL4863168)
Affinity DataIC50: 9.80E+4nMAssay Description:Inhibition of ERAP2 (unknown origin) using R-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570848(CHEMBL4872604)
Affinity DataIC50: 2.19E+5nMAssay Description:Inhibition of ERAP2 (unknown origin) using R-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570848(CHEMBL4872604)
Affinity DataIC50: 2.20E+5nMAssay Description:Inhibition of ERAP2 (unknown origin) using R-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed