Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50013930
TargetPyruvate kinase PKM(Human)
National Institute of Pharmaceutical Education and Research-Ahmedabad

Curated by ChEMBL
LigandPNGBDBM50570977(CHEMBL4878027)
Affinity DataEC50:  5.69E+3nMAssay Description:Activation of PKM2 (unknown origin) by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetPyruvate kinase PKM(Human)
National Institute of Pharmaceutical Education and Research-Ahmedabad

Curated by ChEMBL
LigandPNGBDBM50570976(CHEMBL4866241)
Affinity DataEC50:  6.11E+3nMAssay Description:Activation of PKM2 (unknown origin) by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetPyruvate kinase PKM(Human)
National Institute of Pharmaceutical Education and Research-Ahmedabad

Curated by ChEMBL
LigandPNGBDBM50570975(CHEMBL4859336)
Affinity DataEC50:  7.15E+3nMAssay Description:Activation of PKM2 (unknown origin) by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetPyruvate kinase PKM(Human)
National Institute of Pharmaceutical Education and Research-Ahmedabad

Curated by ChEMBL
LigandPNGBDBM50570978(CHEMBL4868167)
Affinity DataEC50:  8.17E+3nMAssay Description:Activation of PKM2 (unknown origin) by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed