Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50017391
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601516(CHEMBL5181586)
Affinity DataIC50: 80nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601516(CHEMBL5181586)
Affinity DataIC50: 140nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601515(CHEMBL5194499)
Affinity DataIC50: 310nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601518(CHEMBL5173110)
Affinity DataIC50: 740nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601530(CHEMBL5203844)
Affinity DataIC50: 850nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601532(CHEMBL5186486)
Affinity DataIC50: 990nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601517(CHEMBL5181611)
Affinity DataIC50: 990nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601529(CHEMBL5176431)
Affinity DataIC50: 1.05E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601530(CHEMBL5203844)
Affinity DataIC50: 1.18E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601527(CHEMBL5178796)
Affinity DataIC50: 1.22E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601531(CHEMBL5184488)
Affinity DataIC50: 1.54E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601532(CHEMBL5186486)
Affinity DataIC50: 1.59E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601515(CHEMBL5194499)
Affinity DataIC50: 1.85E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601521(CHEMBL5092273)
Affinity DataIC50: 2.15E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601528(CHEMBL5176119)
Affinity DataIC50: 2.87E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601524(CHEMBL5201006)
Affinity DataIC50: 2.99E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601520(CHEMBL5185035)
Affinity DataIC50: 3.29E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601519(CHEMBL5191015)
Affinity DataIC50: 3.93E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601527(CHEMBL5178796)
Affinity DataIC50: 4.18E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601517(CHEMBL5181611)
Affinity DataIC50: 4.30E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601529(CHEMBL5176431)
Affinity DataIC50: 4.92E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601522(CHEMBL5186307)
Affinity DataIC50: 4.95E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601533(CHEMBL5171029)
Affinity DataIC50: 5.21E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601520(CHEMBL5185035)
Affinity DataKd:  6.00E+3nMAssay Description:Binding affinity to recombinant WDR5 (unknown origin) expressed in Escherichia coli BL21 assessed as dissociation constant by isothermal titration ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601518(CHEMBL5173110)
Affinity DataIC50: 8.65E+3nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601519(CHEMBL5191015)
Affinity DataKd:  9.00E+3nMAssay Description:Binding affinity to recombinant WDR5 (unknown origin) expressed in Escherichia coli BL21 assessed as dissociation constant by isothermal titration ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601523(CHEMBL5180413)
Affinity DataKd:  1.10E+4nMAssay Description:Binding affinity to recombinant WDR5 (unknown origin) expressed in Escherichia coli BL21 assessed as dissociation constant by isothermal titration ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601517(CHEMBL5181611)
Affinity DataKd:  1.20E+4nMAssay Description:Binding affinity to recombinant WDR5 (unknown origin) expressed in Escherichia coli BL21 assessed as dissociation constant by isothermal titration ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601522(CHEMBL5186307)
Affinity DataKd:  1.20E+4nMAssay Description:Binding affinity to recombinant WDR5 (unknown origin) expressed in Escherichia coli BL21 assessed as dissociation constant by isothermal titration ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601531(CHEMBL5184488)
Affinity DataIC50: 1.25E+4nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601521(CHEMBL5092273)
Affinity DataIC50: 1.36E+4nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601528(CHEMBL5176119)
Affinity DataIC50: 1.41E+4nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601523(CHEMBL5180413)
Affinity DataIC50: 1.58E+4nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601524(CHEMBL5201006)
Affinity DataIC50: 1.58E+4nMAssay Description:Displacement of N-(4'-((17-(5,5-difluoro-7-(1H-pyrrol-2-yl)-5H-5l4,6l4-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-3-yl)-15-oxo-4,7,10-trioxa-14-azah...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601521(CHEMBL5092273)
Affinity DataKd:  1.80E+4nMAssay Description:Binding affinity to recombinant WDR5 (unknown origin) expressed in Escherichia coli BL21 assessed as dissociation constant by isothermal titration ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601516(CHEMBL5181586)
Affinity DataKd:  2.50E+4nMAssay Description:Binding affinity to recombinant WDR5 (unknown origin) expressed in Escherichia coli BL21 assessed as dissociation constant by isothermal titration ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601524(CHEMBL5201006)
Affinity DataKd:  3.30E+4nMAssay Description:Binding affinity to recombinant WDR5 (unknown origin) expressed in Escherichia coli BL21 assessed as dissociation constant by isothermal titration ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601518(CHEMBL5173110)
Affinity DataKd:  4.10E+4nMAssay Description:Binding affinity to recombinant WDR5 (unknown origin) expressed in Escherichia coli BL21 assessed as dissociation constant by isothermal titration ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601526(CHEMBL5193707)
Affinity DataKd:  9.70E+4nMAssay Description:Binding affinity to recombinant WDR5 (unknown origin) expressed in Escherichia coli BL21 assessed as dissociation constant by isothermal titration ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601515(CHEMBL5194499)
Affinity DataKd:  9.80E+4nMAssay Description:Binding affinity to recombinant WDR5 (unknown origin) expressed in Escherichia coli BL21 assessed as dissociation constant by isothermal titration ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50601525(CHEMBL5186473)
Affinity DataKd:  1.25E+5nMAssay Description:Binding affinity to recombinant WDR5 (unknown origin) expressed in Escherichia coli BL21 assessed as dissociation constant by isothermal titration ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed