Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50015070
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM588477(2-amino-9-[(2S,5S,7R,8R,10S,12aR,14R,15aS)-2,10-di...)
Affinity DataEC50:  172nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Mouse)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582523(CHEMBL5086820)
Affinity DataEC50:  760nMAssay Description:Agonist activity at STING in mouse RAW264.7 cells incubated for 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Mouse)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582522(CHEMBL5092444)
Affinity DataEC50:  500nMAssay Description:Agonist activity at STING in mouse RAW264.7 cells incubated for 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Mouse)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582513(CHEMBL5093161)
Affinity DataEC50:  7.38E+3nMAssay Description:Agonist activity at STING in mouse RAW264.7 cells incubated for 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Mouse)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582523(CHEMBL5086820)
Affinity DataEC50:  280nMAssay Description:Agonist activity at mouse STING in THP-1 dual cells incubated for 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Mouse)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582522(CHEMBL5092444)
Affinity DataEC50:  700nMAssay Description:Agonist activity at mouse STING in THP-1 dual cells incubated for 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Mouse)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582513(CHEMBL5093161)
Affinity DataEC50:  7.16E+3nMAssay Description:Agonist activity at mouse STING in THP-1 dual cells incubated for 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582523(CHEMBL5086820)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at STING KO human THP-1 dual cells incubated for 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582522(CHEMBL5092444)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at STING KO human THP-1 dual cells incubated for 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582513(CHEMBL5093161)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at STING KO human THP-1 dual cells incubated for 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM588530(US11542293, Compound I-5b | 2-amino-9-[(2S,5R,7R,8...)
Affinity DataEC50:  1.91E+3nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM588530(US11542293, Compound I-5b | 2-amino-9-[(2S,5R,7R,8...)
Affinity DataEC50:  1.91E+3nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM588524(US11542293, Compound I-2b | 2-amino-9-[(2S,5R,7R,8...)
Affinity DataEC50:  3.10E+3nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM588589(2-amino-9-[(2S,5R,7R,8R,10S,12aR,14R,15S,15aR,16R)...)
Affinity DataEC50:  30nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM588574(US11542293, Compound I-32b | 2-amino-9-[(2S,5R,7R,...)
Affinity DataEC50:  150nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM588556(US11542293, Compound I-22b | 2-amino-9-[(2S,5R,7R,...)
Affinity DataEC50:  100nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50506263(CHEMBL4465054 | US11401295, Compound 2',3'-cGAMP)
Affinity DataEC50:  50nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM588572(US11542293, Compound I-31b | 2-amino-7-[(2S,5R,7R,...)
Affinity DataEC50:  1.03E+4nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM588537(9-[(2S,5R,7R,8R,10S,12aR,14R,15aS,16R)-16-hydroxy-...)
Affinity DataEC50:  310nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM588568(US11542293, Compound I-30b | 5-amino-3-[(2S,5R,7R,...)
Affinity DataEC50:  80nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582523(CHEMBL5086820)
Affinity DataEC50:  102nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582522(CHEMBL5092444)
Affinity DataEC50:  85nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582521(CHEMBL5094746)
Affinity DataEC50:  3.99E+4nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582520(CHEMBL5084389)
Affinity DataEC50:  4.20E+4nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582519(CHEMBL5073923)
Affinity DataEC50:  4.24E+4nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582518(CHEMBL5081302)
Affinity DataEC50:  890nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582517(CHEMBL5077432)
Affinity DataEC50:  250nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582516(CHEMBL5078624)
Affinity DataEC50:  8.45E+3nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582515(CHEMBL5085601)
Affinity DataEC50:  1.16E+4nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582514(CHEMBL5071799)
Affinity DataEC50:  1.31E+3nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetStimulator of interferon genes protein(Human)
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50582513(CHEMBL5093161)
Affinity DataEC50:  700nMAssay Description:Binding affinity to human STING incubated for 60 mins measured by competitive TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed