Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50014455
TargetAromatase(Human)
Chulabhorn Royal Academy

Curated by ChEMBL
LigandPNGBDBM13061(CHEMBL1444 | 4-[(4-cyanophenyl)(1H-1,2,4-triazol-1...)
Affinity DataIC50: 1nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetAromatase(Human)
Chulabhorn Royal Academy

Curated by ChEMBL
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataIC50: 23nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAromatase(Human)
Chulabhorn Royal Academy

Curated by ChEMBL
LigandPNGBDBM8610(24F2-1,25(OH)D3 | Ketoconazole (k) | KTZ | 1-[4-(4...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetAromatase(Human)
Chulabhorn Royal Academy

Curated by ChEMBL
LigandPNGBDBM50576415(CHEMBL4852023)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetAromatase(Human)
Chulabhorn Royal Academy

Curated by ChEMBL
LigandPNGBDBM50576410(CHEMBL4875917)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetAromatase(Human)
Chulabhorn Royal Academy

Curated by ChEMBL
LigandPNGBDBM50576414(CHEMBL4874928)
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetAromatase(Human)
Chulabhorn Royal Academy

Curated by ChEMBL
LigandPNGBDBM50576413(CHEMBL4863718)
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetAromatase(Human)
Chulabhorn Royal Academy

Curated by ChEMBL
LigandPNGBDBM50576412(CHEMBL4859743)
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetAromatase(Human)
Chulabhorn Royal Academy

Curated by ChEMBL
LigandPNGBDBM50576411(CHEMBL4866633)
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed