Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50013975
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50157526(TCMDC-133606 | CHEMBL586426 | D3RKN_107)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity to BPTF (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50571297(CHEMBL4846718)
Affinity DataKd:  428nMAssay Description:Binding affinity to BPTF (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50571296(CHEMBL4873093)
Affinity DataKd:  71nMAssay Description:Binding affinity to BPTF (unknown origin) by BLI assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50571299(CHEMBL4858897)
Affinity DataKd:  3.55E+4nMAssay Description:Binding affinity to BPTF (unknown origin) by BLI assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50571296(CHEMBL4873093)
Affinity DataIC50: 16nMAssay Description:Inhibition of BPTF in human HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50571296(CHEMBL4873093)
Affinity DataIC50: 30nMAssay Description:Inhibition of BPTF (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetChromatin remodeling regulator CECR2(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50514899(CHEMBL4461619)
Affinity DataIC50: 30nMAssay Description:Inhibition of CECR2 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50514899(CHEMBL4461619)
Affinity DataIC50: 350nMAssay Description:Inhibition of BPTF (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50571298(CHEMBL4846726)
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of N-terminal GST-tagged human recombinant BPTF expressed in Escherichia coli BL21-Codonplus (DE3)-RIPL incubated for 30 mins by HTRF assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed