Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50014805
TargetProtein kinase C epsilon type(Human)
Instituto Nacional De Tecnolog£A Industrial

Curated by ChEMBL
LigandPNGBDBM50107120(2,2-Dimethyl-propionic acid 2-hydroxymethyl-4-[3-i...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]-PDBu from recombinant human PKCepsilon by scintillation counter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Instituto Nacional De Tecnolog£A Industrial

Curated by ChEMBL
LigandPNGBDBM50580096(CHEMBL5078146)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-PDBu from recombinant human PKCalpha at 30 uM by scintillation counter method relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Instituto Nacional De Tecnolog£A Industrial

Curated by ChEMBL
LigandPNGBDBM50107120(2,2-Dimethyl-propionic acid 2-hydroxymethyl-4-[3-i...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]-PDBu from recombinant human PKCalpha by scintillation counter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetProtein kinase C epsilon type(Human)
Instituto Nacional De Tecnolog£A Industrial

Curated by ChEMBL
LigandPNGBDBM50580095(CHEMBL5077090)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]-PDBu from recombinant human PKCepsilon by scintillation counter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Instituto Nacional De Tecnolog£A Industrial

Curated by ChEMBL
LigandPNGBDBM50580095(CHEMBL5077090)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]-PDBu from recombinant human PKCalpha by scintillation counter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed