Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50014233
TargetAromatase(Human)
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50573759(CHEMBL4870604)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human aromatase assessed as reduction in fluorescence intensity using 7-methoxy-4-trifluoromethyl coumarin as a substrate by fluorimetr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetAromatase(Human)
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50573760(CHEMBL4868867)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of human aromatase assessed as reduction in fluorescence intensity using 7-methoxy-4-trifluoromethyl coumarin as a substrate by fluorimetr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetAromatase(Human)
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50210930(CHEMBL3924170)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human aromatase in T47D measured after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetAromatase(Human)
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50573758(CHEMBL4847316)
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of human aromatase assessed as reduction in fluorescence intensity using 7-methoxy-4-trifluoromethyl coumarin as a substrate by fluorimetr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetAromatase(Human)
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50345657(rac-3-((1H-imidazol-1-yl)methyl)-1-(3-tert-butyl-4...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of human aromatase assessed as reduction in fluorescence intensity using 7-methoxy-4-trifluoromethyl coumarin as a substrate by fluorimetr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetAromatase(Human)
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50334280((E)-4-styrylaniline | 4-Styryl-phenylamine | trans...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of human aromatase using dibenzylfluorescein as a substrate preincubated with NADPH regenerating system for 10 mins followed by substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetAromatase(Human)
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM23926(5-[(E)-2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol...)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of human aromatase using dibenzylfluorescein as a substrate preincubated with NADPH regenerating system for 10 mins followed by substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed