Compile Data Set for Download or QSAR
Report error Found 272 Enz. Inhib. hit(s) with all data for entry = 50016825
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597579(CHEMBL5197201)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597589(CHEMBL5209180)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523757(US11136312, Compound MM-I-87)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597576(CHEMBL5180543)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523756(US11136312, Compound MM-I-83)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597581(CHEMBL5183772)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597587(CHEMBL5174969)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597579(CHEMBL5197201)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597581(CHEMBL5183772)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523754(US11136312, Compound MM-I-66)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597590(CHEMBL5185547)
Affinity DataKi:  0.600nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523770(US11136312, Compound SK-I-124)
Affinity DataKi:  0.700nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597590(CHEMBL5185547)
Affinity DataEC50:  0.700nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523770(US11136312, Compound SK-I-124)
Affinity DataEC50:  0.700nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523757(US11136312, Compound MM-I-87)
Affinity DataKi:  0.700nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597580(CHEMBL5179456)
Affinity DataKi:  0.700nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597591(CHEMBL5172814)
Affinity DataKi:  0.700nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597576(CHEMBL5180543)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597587(CHEMBL5174969)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523754(US11136312, Compound MM-I-66)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523767(US11136312, Compound SK-I-91)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597589(CHEMBL5209180)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523755(US11136312, Compound MM-I-72)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523756(US11136312, Compound MM-I-83)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523766(US11136312, Compound SK-I-57)
Affinity DataEC50:  1nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597585(CHEMBL5176083)
Affinity DataEC50:  1nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597585(CHEMBL5176083)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597577(CHEMBL5190056)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597577(CHEMBL5190056)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523760(US11136312, Compound SK-I-22)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523760(US11136312, Compound SK-I-22)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523762(US11136312, Compound SK-I-25)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597586(CHEMBL5173784)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523759(US11136312, Compound SK-I-16)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523759(US11136312, Compound SK-I-16)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523766(US11136312, Compound SK-I-57)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597580(CHEMBL5179456)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523762(US11136312, Compound SK-I-25)
Affinity DataEC50:  2nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597586(CHEMBL5173784)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523761(US11136312, Compound SK-I-23)
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597591(CHEMBL5172814)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597578(CHEMBL5205998)
Affinity DataKi:  2.60nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523764(US11136312, Compound SK-I-55)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523758(US11136312, Compound MM-I-89)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523758(US11136312, Compound MM-I-89)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523763(US11136312, Compound SK-I-53)
Affinity DataKi:  3.10nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM50597578(CHEMBL5205998)
Affinity DataEC50:  3.10nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523738(US11136312, Compound BN-VI-97)
Affinity DataKi:  3.20nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523767(US11136312, Compound SK-I-91)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at recombinant human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSomatostatin receptor type 4(Human)
Southern Illinois University Edwardsville

Curated by ChEMBL
LigandPNGBDBM523765(US11136312, Compound SK-I-56)
Affinity DataKi:  3.30nMAssay Description:Displacement of [125I]-Tyr-SRIF 14 from human SST4 receptor expressed in membrane measured after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
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