Compile Data Set for Download or QSAR
Report error Found 86 Enz. Inhib. hit(s) with all data for entry = 50014945
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM21008((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataEC50:  4.57nMAssay Description:Agonist activity at DOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM21008((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity at DOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM21130(U69,593 | N-methyl-N-(7-(1-pyrrolidinyl)-1-oxaspir...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM21130(U69,593 | N-methyl-N-(7-(1-pyrrolidinyl)-1-oxaspir...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581385(CHEMBL5086601)
Affinity DataEC50:  28nMAssay Description:Agonist activity at DOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581385(CHEMBL5086601)
Affinity DataEC50:  28nMAssay Description:Agonist activity at DOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581385(CHEMBL5086601)
Affinity DataEC50:  29nMAssay Description:Agonist activity at NPFF1R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581385(CHEMBL5086601)
Affinity DataEC50:  29nMAssay Description:Agonist activity at NPFF1R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581389(CHEMBL5091560)
Affinity DataEC50:  38nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581389(CHEMBL5091560)
Affinity DataEC50:  38nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581384(CHEMBL5085455)
Affinity DataEC50:  39nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581384(CHEMBL5085455)
Affinity DataEC50:  39nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50037557(2-{[1-(2-{2-[2-(2-Amino-3-phenyl-propionylamino)-4...)
Affinity DataEC50:  42nMAssay Description:Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50037557(2-{[1-(2-{2-[2-(2-Amino-3-phenyl-propionylamino)-4...)
Affinity DataEC50:  43nMAssay Description:Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581384(CHEMBL5085455)
Affinity DataEC50:  50nMAssay Description:Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581384(CHEMBL5085455)
Affinity DataEC50:  50nMAssay Description:Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581383(CHEMBL5090298)
Affinity DataEC50:  66nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581383(CHEMBL5090298)
Affinity DataEC50:  66nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581389(CHEMBL5091560)
Affinity DataEC50:  71nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataEC50:  71nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581389(CHEMBL5091560)
Affinity DataEC50:  71nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581385(CHEMBL5086601)
Affinity DataEC50:  72nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataEC50:  72nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581385(CHEMBL5086601)
Affinity DataEC50:  73nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581383(CHEMBL5090298)
Affinity DataEC50:  74nMAssay Description:Agonist activity at DOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581383(CHEMBL5090298)
Affinity DataEC50:  74nMAssay Description:Agonist activity at DOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581383(CHEMBL5090298)
Affinity DataEC50:  81nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581383(CHEMBL5090298)
Affinity DataEC50:  81nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581386(CHEMBL5085013)
Affinity DataEC50:  81nMAssay Description:Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581386(CHEMBL5085013)
Affinity DataEC50:  82nMAssay Description:Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581390(CHEMBL5082892)
Affinity DataEC50:  89nMAssay Description:Agonist activity at NPFF1R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581390(CHEMBL5082892)
Affinity DataEC50:  90nMAssay Description:Agonist activity at NPFF1R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581384(CHEMBL5085455)
Affinity DataEC50:  93nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581384(CHEMBL5085455)
Affinity DataEC50:  94nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581389(CHEMBL5091560)
Affinity DataEC50:  95nMAssay Description:Agonist activity at DOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581389(CHEMBL5091560)
Affinity DataEC50:  95nMAssay Description:Agonist activity at DOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581386(CHEMBL5085013)
Affinity DataEC50:  104nMAssay Description:Agonist activity at NPFF1R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581386(CHEMBL5085013)
Affinity DataEC50:  105nMAssay Description:Agonist activity at NPFF1R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581385(CHEMBL5086601)
Affinity DataEC50:  112nMAssay Description:Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581385(CHEMBL5086601)
Affinity DataEC50:  112nMAssay Description:Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581388(CHEMBL5094675)
Affinity DataEC50:  132nMAssay Description:Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581388(CHEMBL5094675)
Affinity DataEC50:  133nMAssay Description:Agonist activity at NPFF2R (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581390(CHEMBL5082892)
Affinity DataEC50:  136nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581388(CHEMBL5094675)
Affinity DataEC50:  138nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581390(CHEMBL5082892)
Affinity DataEC50:  138nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581388(CHEMBL5094675)
Affinity DataEC50:  139nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581386(CHEMBL5085013)
Affinity DataEC50:  166nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581386(CHEMBL5085013)
Affinity DataEC50:  167nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581388(CHEMBL5094675)
Affinity DataEC50:  168nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50581388(CHEMBL5094675)
Affinity DataEC50:  170nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
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