Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50014560
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506458(CHEMBL4576115)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human recombinant CSF1R using ATP/Ulight-TK peptide incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506469(CHEMBL4438121)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human recombinant CSF1R using ATP/Ulight-TK peptide incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506459(CHEMBL4517659)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human recombinant CSF1R using ATP/Ulight-TK peptide incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506450(CHEMBL4553298)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human recombinant CSF1R using ATP/Ulight-TK peptide incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506470(CHEMBL4589346)
Affinity DataIC50: 3nMAssay Description:Inhibition of human recombinant CSF1R using ATP/Ulight-TK peptide incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506460(CHEMBL4467948)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of human recombinant CSF1R using ATP/Ulight-TK peptide incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506460(CHEMBL4467948)
Affinity DataIC50: 7nMAssay Description:Inhibition of human full length recombinant LYN by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506460(CHEMBL4467948)
Affinity DataIC50: 7nMAssay Description:Inhibition of human recombinant ABL1 using ATP/Ulight-TK peptide incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577409(CHEMBL4854948)
Affinity DataIC50: 8nMAssay Description:Inhibition of human recombinant CSF1R using ATP/Ulight-TK peptide incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50322535(3-[2-(Imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-meth...)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of human recombinant CSF1R using ATP/Ulight-TK peptide incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase HCK(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577406(CHEMBL4862806)
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant HCK (230 to 497) by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577406(CHEMBL4862806)
Affinity DataIC50: 9nMAssay Description:Inhibition of human full length recombinant LYN by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506460(CHEMBL4467948)
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant CSF1R using ATP/Ulight-TK peptide at 50 nM incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577406(CHEMBL4862806)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant Src (1-530) by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50177716(CHEMBL3813873 | US11679110, Compound Pexidartinib ...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant CSF1R using ATP/Ulight-TK peptide incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase ABL1(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577406(CHEMBL4862806)
Affinity DataIC50: 22nMAssay Description:Inhibition of human recombinant ABL1 using ATP/Ulight-TK peptide incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577408(CHEMBL4850154)
Affinity DataIC50: 22nMAssay Description:Inhibition of human recombinant CSF1R using ATP/Ulight-TK peptide incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577407(CHEMBL4854116)
Affinity DataIC50: 24nMAssay Description:Inhibition of human recombinant CSF1R using ATP/Ulight-TK peptide incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506460(CHEMBL4467948)
Affinity DataIC50: 29nMAssay Description:Inhibition of human full length recombinant LCK by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577410(CHEMBL4869362)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant CSF1R using ATP/Ulight-TK peptide incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Fgr(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577406(CHEMBL4862806)
Affinity DataIC50: 41nMAssay Description:Inhibition of human recombinant FGR (456 to 770) radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577406(CHEMBL4862806)
Affinity DataIC50: 48nMAssay Description:Inhibition of human recombinant CSF1R using ATP/Ulight-TK peptide at 50 nM incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577406(CHEMBL4862806)
Affinity DataIC50: 48nMAssay Description:Inhibition of human recombinant CSF1R using ATP/Ulight-TK peptide incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Fyn(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577406(CHEMBL4862806)
Affinity DataIC50: 56nMAssay Description:Inhibition of human full length recombinant Fyn by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Blk(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577406(CHEMBL4862806)
Affinity DataIC50: 56nMAssay Description:Inhibition of human full length recombinant BLK by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase HCK(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506460(CHEMBL4467948)
Affinity DataIC50: 57nMAssay Description:Inhibition of human recombinant HCK (230 to 497) by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Yes(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577406(CHEMBL4862806)
Affinity DataIC50: 95nMAssay Description:Inhibition of human full length recombinant Yes by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577406(CHEMBL4862806)
Affinity DataIC50: 101nMAssay Description:Inhibition of human full length recombinant LCK by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Srms(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577406(CHEMBL4862806)
Affinity DataIC50: 114nMAssay Description:Inhibition of human SRMS by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCytoplasmic tyrosine-protein kinase BMX(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577406(CHEMBL4862806)
Affinity DataIC50: 126nMAssay Description:Inhibition of human full length recombinant Bmx by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506460(CHEMBL4467948)
Affinity DataIC50: 163nMAssay Description:Inhibition of human recombinant Src (1-530) by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCytoplasmic tyrosine-protein kinase BMX(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577406(CHEMBL4862806)
Affinity DataIC50: 185nMAssay Description:Inhibition of human recombinant Txk (256 to end) by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase CSK(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50577406(CHEMBL4862806)
Affinity DataIC50: 187nMAssay Description:Inhibition of human full length recombinant CSK by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Fyn(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506460(CHEMBL4467948)
Affinity DataIC50: 307nMAssay Description:Inhibition of human full length recombinant Fyn by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase CSK(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506460(CHEMBL4467948)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human full length recombinant CSK by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Blk(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506460(CHEMBL4467948)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human full length recombinant BLK by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Fgr(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506460(CHEMBL4467948)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant FGR (456 to 770) radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Srms(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506460(CHEMBL4467948)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human SRMS by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Yes(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506460(CHEMBL4467948)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human full length recombinant Yes by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCytoplasmic tyrosine-protein kinase BMX(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506460(CHEMBL4467948)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human full length recombinant Bmx by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCytoplasmic tyrosine-protein kinase BMX(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50506460(CHEMBL4467948)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant Txk (256 to end) by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed