Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50014717
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.70nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 5.10nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 5.60nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 7.60nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 8.70nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 9.70nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 394nMAssay Description:Inhibition of recombinant human c-Kit assessed as luminescence using poly (4:1 Glu, Tyr) peptide as substrate incubated for 2 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 496nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.63E+3nMAssay Description:Inhibition of recombinant human c-Kit assessed as luminescence using poly (4:1 Glu, Tyr) peptide as substrate incubated for 2 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.98E+3nMAssay Description:Inhibition of recombinant human c-Kit assessed as luminescence using poly (4:1 Glu, Tyr) peptide as substrate incubated for 2 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.43E+3nMAssay Description:Inhibition of recombinant human PDGFRalpha assessed as luminescence using poly (4:1 Glu, Tyr) peptide as substrate incubated for 1 hr by ADP-Glo assa...More data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.66E+3nMAssay Description:Inhibition of recombinant human c-Kit assessed as luminescence using poly (4:1 Glu, Tyr) peptide as substrate incubated for 2 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 5.24E+3nMAssay Description:Inhibition of recombinant human PDGFRalpha assessed as luminescence using poly (4:1 Glu, Tyr) peptide as substrate incubated for 1 hr by ADP-Glo assa...More data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of recombinant human c-Kit assessed as luminescence using poly (4:1 Glu, Tyr) peptide as substrate incubated for 2 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 7.44E+3nMAssay Description:Inhibition of recombinant human c-Kit assessed as luminescence using poly (4:1 Glu, Tyr) peptide as substrate incubated for 2 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 8.41E+3nMAssay Description:Inhibition of recombinant human c-Kit assessed as luminescence using poly (4:1 Glu, Tyr) peptide as substrate incubated for 2 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 9.45E+3nMAssay Description:Inhibition of recombinant human PDGFRalpha assessed as luminescence using poly (4:1 Glu, Tyr) peptide as substrate incubated for 1 hr by ADP-Glo assa...More data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human c-Kit assessed as luminescence using poly (4:1 Glu, Tyr) peptide as substrate incubated for 2 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human PDGFRalpha assessed as luminescence using poly (4:1 Glu, Tyr) peptide as substrate incubated for 1 hr by ADP-Glo assa...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human PDGFRalpha assessed as luminescence using poly (4:1 Glu, Tyr) peptide as substrate incubated for 1 hr by ADP-Glo assa...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Johns Hopkins University School of Medicine
Curated by ChEMBL
Johns Hopkins University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human His-tagged c-Abl kinase assessed as luminescence incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair




































