Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50014725
TargetHistone deacetylase 6(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50380399(CHEMBL2018302 | US8748451, 6 | Tubastatin A | US92...)
Affinity DataIC50: 15nMAssay Description:Inhibition of recombiant human HDAC6 using fluorogenic HDAC substrate 3 measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombiant human HDAC6 using fluorogenic HDAC substrate 3 measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579532(CHEMBL4867598)
Affinity DataIC50: 27nMAssay Description:Inhibition of full length human CDK6 (1 to 326 end residues)/N-terminal GST-fusion tagged CyclinD3 (1 to 292 residues) expressed in baculovirus expre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579532(CHEMBL4867598)
Affinity DataIC50: 61nMAssay Description:Inhibition of full length human CDK2 (1 to 298 end residues)/N-terminal GST-tagged CyclinA2 (1 to 432 residues) expressed in baculovirus expression s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579533(CHEMBL4859978)
Affinity DataIC50: 68nMAssay Description:Inhibition of full length human CDK6 (1 to 326 end residues)/N-terminal GST-fusion tagged CyclinD3 (1 to 292 residues) expressed in baculovirus expre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 83nMAssay Description:Inhibition of HDAC8 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 1(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 88nMAssay Description:Inhibition of HDAC1 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 90nMAssay Description:Inhibition of C-terminal His-tagged recombinant human HDAC3 (1 to 428 residues)/N-terminal GST-tagged recombinant human NCoR2 (395 to 489 residues) c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579533(CHEMBL4859978)
Affinity DataIC50: 119nMAssay Description:Inhibition of full length human CDK2 (1 to 298 end residues)/N-terminal GST-tagged CyclinA2 (1 to 432 residues) expressed in baculovirus expression s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579532(CHEMBL4867598)
Affinity DataIC50: 129nMAssay Description:Inhibition of recombiant human HDAC6 using fluorogenic HDAC substrate 3 measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 200nMAssay Description:Inhibition of HDAC2 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579532(CHEMBL4867598)
Affinity DataIC50: 276nMAssay Description:Inhibition of full length human CDK4 (1 to 303 residues)/N-terminal GST-fusion tagged CyclinD3 (1 to 292 residues) expressed in baculovirus expressio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50380399(CHEMBL2018302 | US8748451, 6 | Tubastatin A | US92...)
Affinity DataIC50: 854nMAssay Description:Inhibition of HDAC8 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579534(CHEMBL4877598)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of full length human CDK6 (1 to 326 end residues)/N-terminal GST-fusion tagged CyclinD3 (1 to 292 residues) expressed in baculovirus expre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579534(CHEMBL4877598)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of full length human CDK2 (1 to 298 end residues)/N-terminal GST-tagged CyclinA2 (1 to 432 residues) expressed in baculovirus expression s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579534(CHEMBL4877598)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of full length human CDK4 (1 to 303 residues)/N-terminal GST-fusion tagged CyclinD3 (1 to 292 residues) expressed in baculovirus expressio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579534(CHEMBL4877598)
Affinity DataIC50: 1.87E+3nMAssay Description:Inhibition of recombiant human HDAC6 using fluorogenic HDAC substrate 3 measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579533(CHEMBL4859978)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombiant human HDAC6 using fluorogenic HDAC substrate 3 measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 7(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579532(CHEMBL4867598)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC7 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 7(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579533(CHEMBL4859978)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC7 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 7(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579534(CHEMBL4877598)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC7 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 7(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50380399(CHEMBL2018302 | US8748451, 6 | Tubastatin A | US92...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC7 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 7(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC7 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 8(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579532(CHEMBL4867598)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC8 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579533(CHEMBL4859978)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC8 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579534(CHEMBL4877598)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC8 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 9(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579532(CHEMBL4867598)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human HDAC9 measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 9(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579533(CHEMBL4859978)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human HDAC9 measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579532(CHEMBL4867598)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of C-terminal His-tagged recombinant human HDAC3 (1 to 428 residues)/N-terminal GST-tagged recombinant human NCoR2 (395 to 489 residues) c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579533(CHEMBL4859978)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of C-terminal His-tagged recombinant human HDAC3 (1 to 428 residues)/N-terminal GST-tagged recombinant human NCoR2 (395 to 489 residues) c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50380399(CHEMBL2018302 | US8748451, 6 | Tubastatin A | US92...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of C-terminal His-tagged recombinant human HDAC3 (1 to 428 residues)/N-terminal GST-tagged recombinant human NCoR2 (395 to 489 residues) c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579532(CHEMBL4867598)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC4 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579533(CHEMBL4859978)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC4 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50380399(CHEMBL2018302 | US8748451, 6 | Tubastatin A | US92...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC4 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC4 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579532(CHEMBL4867598)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC5 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579533(CHEMBL4859978)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC5 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50380399(CHEMBL2018302 | US8748451, 6 | Tubastatin A | US92...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC5 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC5 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579532(CHEMBL4867598)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC1 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579533(CHEMBL4859978)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC1 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50380399(CHEMBL2018302 | US8748451, 6 | Tubastatin A | US92...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC1 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579532(CHEMBL4867598)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC2 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579533(CHEMBL4859978)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC2 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50380399(CHEMBL2018302 | US8748451, 6 | Tubastatin A | US92...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC2 (unknown origin) measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 9(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50380399(CHEMBL2018302 | US8748451, 6 | Tubastatin A | US92...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human HDAC9 measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 9(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human HDAC9 measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 11(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579532(CHEMBL4867598)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human HDAC11 measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 11(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579533(CHEMBL4859978)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human HDAC11 measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
TargetHistone deacetylase 11(Human)
Guizhou Medical University

Curated by ChEMBL
LigandPNGBDBM50579534(CHEMBL4877598)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human HDAC11 measured after 30 mins by fluorescence microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2022
Entry Details Article
PubMed
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