Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50018428
TargetTrace amine-associated receptor 1(Human)
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataEC50: 140nMAssay Description:Agonist activity at human TAAR1More data for this Ligand-Target Pair
3D Structure (crystal)Target5-hydroxytryptamine receptor 1A(Human)
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataEC50: 2.30E+3nMAssay Description:Agonist activity at 5HT1A (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+4nMAssay Description:Agonist activity at D2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Positive allosteric modulator activity at human M4 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Positive allosteric modulator activity at rat M4 receptor by FLIPR assayMore data for this Ligand-Target Pair
TargetHigh affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A(Human)
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of human PDE9A expressed in Escherichia coli DH10 by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+4nMAssay Description:Agonist activity at D2 (unknown origin) by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
