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Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50016604
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596039(CHEMBL5186555)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596040(CHEMBL5193065)
Affinity DataIC50: 4.80nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596035(CHEMBL5189611)
Affinity DataIC50: 6.10nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596034(CHEMBL5175004)
Affinity DataIC50: 6.70nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596030(CHEMBL5191983)
Affinity DataIC50: 8.70nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596045(CHEMBL5172530)
Affinity DataIC50: 9.20nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596031(CHEMBL5204942)
Affinity DataIC50: 9.30nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596037(CHEMBL5180780)
Affinity DataIC50: 9.70nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596048(CHEMBL5186024)
Affinity DataIC50: 9.80nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596041(CHEMBL5174678)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596044(CHEMBL5198913)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596028(CHEMBL5170675)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596047(CHEMBL5184355)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596036(CHEMBL5177634)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596043(CHEMBL5191737)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596049(CHEMBL5186756)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596026(CHEMBL5190464)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596029(CHEMBL5177972)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596042(CHEMBL5180500)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596046(CHEMBL5192666)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596032(CHEMBL5173454)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596038(CHEMBL5186266)
Affinity DataIC50: 28nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596033(CHEMBL5191340)
Affinity DataIC50: 33nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596027(CHEMBL5175099)
Affinity DataIC50: 35nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50596050(CHEMBL5198960)
Affinity DataIC50: 42nMAssay Description:Antagonist activity at human P2Y14R expressed in human HEK293 cells assessed as inhibition of cAMP level incubated for 30 mins by cAMP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed