Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50014351
TargetEndothelial PAS domain-containing protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50575225(CHEMBL4877680)
Affinity DataEC50:  5.62E+3nMAssay Description:Agonist activity at HIF-2alpha (unknown origin) expressed in 786-O cells measured after 24 hrs by HRE based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50575226(CHEMBL4853289)
Affinity DataEC50:  1.68E+3nMAssay Description:Agonist activity at HIF-2alpha (unknown origin) expressed in 786-O cells measured after 24 hrs by HRE based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50575227(CHEMBL4857622)
Affinity DataEC50:  1.35E+3nMAssay Description:Agonist activity at HIF-2alpha (unknown origin) expressed in 786-O cells measured after 24 hrs by HRE based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50575228(CHEMBL4879236)
Affinity DataEC50:  1.76E+3nMAssay Description:Agonist activity at HIF-2alpha (unknown origin) expressed in 786-O cells measured after 24 hrs by HRE based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50575229(CHEMBL4868087)
Affinity DataEC50:  2.98E+3nMAssay Description:Agonist activity at HIF-2alpha (unknown origin) expressed in 786-O cells measured after 24 hrs by HRE based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50575230(CHEMBL4846319)
Affinity DataEC50:  2.92E+3nMAssay Description:Agonist activity at HIF-2alpha (unknown origin) expressed in 786-O cells measured after 24 hrs by HRE based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50575231(CHEMBL4869108)
Affinity DataEC50:  490nMAssay Description:Agonist activity at HIF-2alpha (unknown origin) expressed in 786-O cells measured after 24 hrs by HRE based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50575232(CHEMBL4862826)
Affinity DataEC50:  1.49E+3nMAssay Description:Agonist activity at HIF-2alpha (unknown origin) expressed in 786-O cells measured after 24 hrs by HRE based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50575233(CHEMBL4874183)
Affinity DataEC50:  1.61E+3nMAssay Description:Agonist activity at HIF-2alpha (unknown origin) expressed in 786-O cells measured after 24 hrs by HRE based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50575234(CHEMBL4849634)
Affinity DataEC50:  1.08E+3nMAssay Description:Agonist activity at HIF-2alpha (unknown origin) expressed in 786-O cells measured after 24 hrs by HRE based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50575235(CHEMBL4878756)
Affinity DataEC50:  1.12E+3nMAssay Description:Agonist activity at HIF-2alpha (unknown origin) expressed in 786-O cells measured after 24 hrs by HRE based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed