Compile Data Set for Download or QSAR
Report error Found 85 Enz. Inhib. hit(s) with all data for entry = 50015464
TargetKappa-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586821(CHEMBL5089012)
Affinity DataIC50: 0.537nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586821(CHEMBL5089012)
Affinity DataIC50: 0.692nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586820(CHEMBL5094499)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586817(CHEMBL5091642)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586819(CHEMBL5086370)
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586818(CHEMBL5078669)
Affinity DataIC50: 1.60nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586820(CHEMBL5094499)
Affinity DataIC50: 1.90nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586816(CHEMBL5081245)
Affinity DataIC50: 2.30nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586823(CHEMBL5090705)
Affinity DataIC50: 2.60nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586821(CHEMBL5089012)
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586815(CHEMBL5083183)
Affinity DataIC50: 4.60nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586819(CHEMBL5086370)
Affinity DataIC50: 4.70nMAssay Description:Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM21123(Enkephalin Amide | (2S)-2-{2-[(2R)-2-[(2S)-2-amino...)
Affinity DataIC50: 5.80nMAssay Description:Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586819(CHEMBL5086370)
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586818(CHEMBL5078669)
Affinity DataIC50: 7.60nMAssay Description:Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586822(CHEMBL5077561)
Affinity DataIC50: 7.80nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586817(CHEMBL5091642)
Affinity DataIC50: 8.10nMAssay Description:Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586816(CHEMBL5081245)
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586820(CHEMBL5094499)
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586815(CHEMBL5083183)
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586823(CHEMBL5090705)
Affinity DataIC50: 23nMAssay Description:Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586818(CHEMBL5078669)
Affinity DataIC50: 24nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586822(CHEMBL5077561)
Affinity DataIC50: 78nMAssay Description:Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586817(CHEMBL5091642)
Affinity DataIC50: 83nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586823(CHEMBL5090705)
Affinity DataIC50: 98nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586822(CHEMBL5077561)
Affinity DataIC50: 123nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586815(CHEMBL5083183)
Affinity DataIC50: 182nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586816(CHEMBL5081245)
Affinity DataIC50: 191nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM21123(Enkephalin Amide | (2S)-2-{2-[(2R)-2-[(2S)-2-amino...)
Affinity DataIC50: 224nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM21123(Enkephalin Amide | (2S)-2-{2-[(2R)-2-[(2S)-2-amino...)
Affinity DataIC50: 724nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586821(CHEMBL5089012)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586821(CHEMBL5089012)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586820(CHEMBL5094499)
Affinity DataKi:  0.530nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586820(CHEMBL5094499)
Affinity DataKi:  0.540nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586817(CHEMBL5091642)
Affinity DataKi:  0.570nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586819(CHEMBL5086370)
Affinity DataKi:  0.580nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586818(CHEMBL5078669)
Affinity DataKi:  0.740nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586816(CHEMBL5081245)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586823(CHEMBL5090705)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586821(CHEMBL5089012)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586819(CHEMBL5086370)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586819(CHEMBL5086370)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586815(CHEMBL5083183)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM21124((2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM21123(Enkephalin Amide | (2S)-2-{2-[(2R)-2-[(2S)-2-amino...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM35229(Desmethylimipramine | 3-(10,11-dihydro-5H-dibenzo[...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-Nisoxetine from human NET expressed in HEK cell membrane assessed as inhibition constant by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMu-type opioid receptor(Rat)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586818(CHEMBL5078669)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586817(CHEMBL5091642)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]-DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM50586822(CHEMBL5077561)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells assessed as inhibition constant by radioligand binding as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of The Punjab

Curated by ChEMBL
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]-WIN35428 from human DAT expressed in HEK cell membrane assessed as inhibition constant by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
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