Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50015032
TargetEpithelial discoidin domain-containing receptor 1(Human)
Bytedance Ai Lab

Curated by ChEMBL
LigandPNGBDBM50582160(CHEMBL5072982)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human DDR1 (492 to end residues) using KKKSPGEYVNIEFG as substrate incubated for 40 mins in presence of [gamma33P]ATP by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Bytedance Ai Lab

Curated by ChEMBL
LigandPNGBDBM50582161(CHEMBL5076889)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human DDR1 (492 to end residues) using KKKSPGEYVNIEFG as substrate incubated for 40 mins in presence of [gamma33P]ATP by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Bytedance Ai Lab

Curated by ChEMBL
LigandPNGBDBM50582159(CHEMBL5082740)
Affinity DataIC50: 28nMAssay Description:Inhibition of recombinant human DDR1 (492 to end residues) using KKKSPGEYVNIEFG as substrate incubated for 40 mins in presence of [gamma33P]ATP by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Bytedance Ai Lab

Curated by ChEMBL
LigandPNGBDBM50582161(CHEMBL5076889)
Affinity DataEC50:  34nMAssay Description:Inhibition of DDR1 in human THP-1 cells assessed as reduction in collagen induced DDR1 autophosphorylation by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Bytedance Ai Lab

Curated by ChEMBL
LigandPNGBDBM50582163(CHEMBL5094596)
Affinity DataIC50: 43nMAssay Description:Inhibition of recombinant human DDR1 (492 to end residues) using KKKSPGEYVNIEFG as substrate incubated for 40 mins in presence of [gamma33P]ATP by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Bytedance Ai Lab

Curated by ChEMBL
LigandPNGBDBM50582162(CHEMBL5072528)
Affinity DataIC50: 49nMAssay Description:Inhibition of recombinant human DDR1 (492 to end residues) using KKKSPGEYVNIEFG as substrate incubated for 40 mins in presence of [gamma33P]ATP by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Bytedance Ai Lab

Curated by ChEMBL
LigandPNGBDBM50582164(CHEMBL5088050)
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant human DDR1 (492 to end residues) using KKKSPGEYVNIEFG as substrate incubated for 40 mins in presence of [gamma33P]ATP by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Bytedance Ai Lab

Curated by ChEMBL
LigandPNGBDBM50582160(CHEMBL5072982)
Affinity DataEC50:  115nMAssay Description:Inhibition of DDR1 in human THP-1 cells assessed as reduction in collagen induced DDR1 autophosphorylation by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Bytedance Ai Lab

Curated by ChEMBL
LigandPNGBDBM50582167(CHEMBL5084624)
Affinity DataIC50: 164nMAssay Description:Inhibition of recombinant human DDR1 (492 to end residues) using KKKSPGEYVNIEFG as substrate incubated for 40 mins in presence of [gamma33P]ATP by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Bytedance Ai Lab

Curated by ChEMBL
LigandPNGBDBM50582168(CHEMBL5075627)
Affinity DataIC50: 235nMAssay Description:Inhibition of recombinant human DDR1 (492 to end residues) using KKKSPGEYVNIEFG as substrate incubated for 40 mins in presence of [gamma33P]ATP by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Bytedance Ai Lab

Curated by ChEMBL
LigandPNGBDBM50582165(CHEMBL5083118)
Affinity DataIC50: 376nMAssay Description:Inhibition of recombinant human DDR1 (492 to end residues) using KKKSPGEYVNIEFG as substrate incubated for 40 mins in presence of [gamma33P]ATP by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Bytedance Ai Lab

Curated by ChEMBL
LigandPNGBDBM50582166(CHEMBL5081927)
Affinity DataIC50: 826nMAssay Description:Inhibition of recombinant human DDR1 (492 to end residues) using KKKSPGEYVNIEFG as substrate incubated for 40 mins in presence of [gamma33P]ATP by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed