Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50015471
TargetMicrotubule-associated protein tau(Human)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586984(CHEMBL5084771)
Affinity DataIC50: 3.10nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586985(CHEMBL5082735)
Affinity DataIC50: 3.5nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586972(CHEMBL5088921)
Affinity DataIC50: 4.90nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Mouse)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586985(CHEMBL5082735)
Affinity DataIC50: 7.80nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586975(CHEMBL5081662)
Affinity DataIC50: 16nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586986(CHEMBL5091624)
Affinity DataIC50: 18nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586979(CHEMBL5084917)
Affinity DataIC50: 36nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Mouse)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586984(CHEMBL5084771)
Affinity DataIC50: 51nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586982(CHEMBL5083649)
Affinity DataIC50: 70nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586973(CHEMBL5077904)
Affinity DataIC50: 82nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586974(CHEMBL5090407)
Affinity DataIC50: 116nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586978(CHEMBL5080178)
Affinity DataIC50: 260nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586980(CHEMBL5081126)
Affinity DataIC50: 310nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586977(CHEMBL5081957)
Affinity DataIC50: 344nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586981(CHEMBL5094590)
Affinity DataIC50: 559nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586976(CHEMBL5092563)
Affinity DataIC50: 732nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586983(CHEMBL5091757)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]PI-2620 from Tau in human brain homogenate incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Mouse)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586972(CHEMBL5088921)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Mouse)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586973(CHEMBL5077904)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Mouse)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586974(CHEMBL5090407)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Mouse)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586975(CHEMBL5081662)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Mouse)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586976(CHEMBL5092563)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Mouse)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586977(CHEMBL5081957)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Mouse)
Ac Immune

Curated by ChEMBL
LigandPNGBDBM50586986(CHEMBL5091624)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed