Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50014906
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581017(CHEMBL5081158)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581003(CHEMBL5084431)
Affinity DataEC50:  70nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50526409(CHEMBL4522365)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581005(CHEMBL5093542)
Affinity DataEC50:  238nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581006(CHEMBL5076246)
Affinity DataEC50:  56nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581007(CHEMBL5082272)
Affinity DataEC50:  98nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581008(CHEMBL5078386)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581009(CHEMBL5094670)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581010(CHEMBL5072593)
Affinity DataEC50:  7.70nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581011(CHEMBL5089682)
Affinity DataEC50:  855nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581012(CHEMBL5077251)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581013(CHEMBL5072912)
Affinity DataEC50:  273nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581014(CHEMBL5078074)
Affinity DataEC50:  73nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581015(CHEMBL5094396)
Affinity DataEC50:  53nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581016(CHEMBL5083969)
Affinity DataEC50:  5.60nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581004(CHEMBL5075697)
Affinity DataEC50:  67nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581018(CHEMBL5084331)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581019(CHEMBL5089949)
Affinity DataEC50:  3.10nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581020(CHEMBL5094669)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50526409(CHEMBL4522365)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as beta arrestin-2 recruitment measured after 4 hrs by beta-galactosidase ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50526408(CHEMBL4586446)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as beta arrestin-2 recruitment measured after 4 hrs by beta-galactosidase ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581017(CHEMBL5081158)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as beta arrestin-2 recruitment measured after 4 hrs by beta-galactosidase ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581019(CHEMBL5089949)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as beta arrestin-2 recruitment measured after 4 hrs by beta-galactosidase ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50526409(CHEMBL4522365)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at human RXFP4 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRelaxin-3 receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581010(CHEMBL5072593)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at human RXFP4 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581016(CHEMBL5083969)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human RXFP4 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581017(CHEMBL5081158)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at human RXFP4 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581018(CHEMBL5084331)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human RXFP4 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581019(CHEMBL5089949)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human RXFP4 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581020(CHEMBL5094669)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human RXFP4 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50580987(CHEMBL5089792)
Affinity DataEC50:  2.82E+3nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50580975(CHEMBL5084645)
Affinity DataEC50:  6.94E+3nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50580976(CHEMBL5081867)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50580977(CHEMBL5078875)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50580978(CHEMBL5077878)
Affinity DataEC50:  7.44E+3nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50580979(CHEMBL5082989)
Affinity DataEC50:  647nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50580980(CHEMBL5074457)
Affinity DataEC50:  1.68E+3nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50580981(CHEMBL5080062)
Affinity DataEC50:  4.75E+3nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50580982(CHEMBL5080322)
Affinity DataEC50:  4.95E+3nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50580983(CHEMBL5084549)
Affinity DataEC50:  3.21E+3nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50580984(CHEMBL5090612)
Affinity DataEC50:  1.36E+3nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50580985(CHEMBL5084224)
Affinity DataEC50:  3.47E+3nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50580986(CHEMBL5090147)
Affinity DataEC50:  2.79E+3nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581002(CHEMBL5078678)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50580988(CHEMBL5091447)
Affinity DataEC50:  5.24E+3nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50580990(CHEMBL5080373)
Affinity DataEC50:  312nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50526408(CHEMBL4586446)
Affinity DataEC50:  306nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581001(CHEMBL5075621)
Affinity DataEC50:  1.28E+3nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50581000(CHEMBL5073543)
Affinity DataEC50:  797nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50580999(CHEMBL5089400)
Affinity DataEC50:  224nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
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