Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50015663
TargetAmine oxidase [flavin-containing] A(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 0.610nMAssay Description:Inhibition of human full length recombinant MAO-A expressed in insect cells using kynuramine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetAmine oxidase [flavin-containing] B(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588335(CHEMBL5170163)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of human full length recombinant MAO-B expressed in insect cells using kynuramine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50: 20nMAssay Description:Inhibition of human HDAC6 (379 to 382 residues) using RHKKAc as flurogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50: 133nMAssay Description:Inhibition of human HDAC3 (379 to 382 residues) using RHKKAc as flurogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetHistone deacetylase 8(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50: 210nMAssay Description:Inhibition of human HDAC8 (379 to 382 residues) using RHKAcKAc as flurogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetPolyamine deacetylase HDAC10(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50: 374nMAssay Description:Inhibition of human HDAC10 using Ac-Spermidine-AMC as flurogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50: 673nMAssay Description:Inhibition of human HDAC1 (379 to 382 residues) using RHKKAc as flurogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50: 790nMAssay Description:Inhibition of human full length recombinant MAO-A expressed in insect cells using kynuramine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetHistone deacetylase 2(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50: 1.54E+3nMAssay Description:Inhibition of human HDAC2 (379 to 382 residues) using RHKKAc as flurogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetHistone deacetylase 4(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as flurogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetHistone deacetylase 7(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human HDAC7 using Boc-Lys(trifluoroacetyl)-AMC as flurogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetHistone deacetylase 9(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human HDAC9 using Boc-Lys(trifluoroacetyl)-AMC as flurogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetHistone deacetylase 5(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50: 1.34E+4nMAssay Description:Inhibition of human HDAC5 using Boc-Lys(trifluoroacetyl)-AMC as flurogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibition of human full length recombinant MAO-B expressed in insect cells using kynuramine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed