Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50018308
TargetRyanodine receptor 2(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50421670(CHEMBL5188974)
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of RyR2 in Casq2 gene knockout mouse cardiomyocytes assessed as reduction in calcium sparks frequency incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetRyanodine receptor 2(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50421669(CHEMBL5180539)
Affinity DataIC50: 3.88E+3nMAssay Description:Inhibition of RyR2 in Casq2 gene knockout mouse cardiomyocytes assessed as reduction in calcium sparks frequency incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed