Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50017596
TargetHistone deacetylase 6(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 7.30nMAssay Description:Inhibition of HDAC6 (unknown origin) using trypsin and Ac-peptide as substratesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50603205(CHEMBL5172182)
Affinity DataIC50: 16nMAssay Description:Inhibition of HDAC6 (unknown origin) using trypsin and Ac-peptide as substratesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 17nMAssay Description:Inhibition of HDAC1 (unknown origin) using trypsin and Ac-peptide as substratesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50603205(CHEMBL5172182)
Affinity DataIC50: 20nMAssay Description:Inhibition of HDAC1 (unknown origin) using trypsin and Ac-peptide as substratesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 22nMAssay Description:Inhibition of HDAC2 (unknown origin) using trypsin and Ac-peptide as substratesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50603205(CHEMBL5172182)
Affinity DataIC50: 27nMAssay Description:Inhibition of HDAC2 (unknown origin) using trypsin and Ac-peptide as substratesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50446481(CHEMBL3110004 | US10011611, TMP269 | US10722597, C...)
Affinity DataIC50: 318nMAssay Description:Inhibition of HDAC4 (unknown origin) using trypsin and Ac-peptide as substratesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetEgl nine homolog 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50431015(CHEMBL2338329 | US9115085, Compound A Form A | US9...)
Affinity DataIC50: 520nMAssay Description:Inhibition of PHD2 (unknown origin) measured by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetEgl nine homolog 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50603205(CHEMBL5172182)
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of PHD2 (unknown origin) measured by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetHistone deacetylase 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50603205(CHEMBL5172182)
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of HDAC4 (unknown origin) using trypsin and Ac-peptide as substratesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed