Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50015253
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584668(CHEMBL5089414)
Affinity DataIC50: 33nMAssay Description:Inhibition of recombinant human N-terminal His-tagged ALOX15 expressed in Escherichia coli Rosetta2(DE3)pLysS using linoleic acid as substrate by spe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584668(CHEMBL5089414)
Affinity DataIC50: 40nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using linoleic acid as substrate by spectrophotometric assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584669(CHEMBL5089447)
Affinity DataIC50: 47nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using linoleic acid as substrate by spectrophotometric assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584663(CHEMBL5090671)
Affinity DataIC50: 420nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using linoleic acid as substrate by spectrophotometric assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584666(CHEMBL5070865)
Affinity DataIC50: 540nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using linoleic acid as substrate by spectrophotometric assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584665(CHEMBL5086474)
Affinity DataIC50: 630nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using linoleic acid as substrate by spectrophotometric assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584668(CHEMBL5089414)
Affinity DataIC50: 650nMAssay Description:Inhibition of recombinant human N-terminal His-tagged ALOX15 expressed in Escherichia coli Rosetta2(DE3)pLysS using arachidonic acid as substrate by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584669(CHEMBL5089447)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using arachidonic acid as substrate by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584662(CHEMBL5088464)
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using linoleic acid as substrate by spectrophotometric assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584667(CHEMBL5080282)
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using linoleic acid as substrate by spectrophotometric assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584668(CHEMBL5089414)
Affinity DataIC50: 2.06E+3nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using arachidonic acid as substrate by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584667(CHEMBL5080282)
Affinity DataIC50: 2.79E+3nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using arachidonic acid as substrate by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584664(CHEMBL5070746)
Affinity DataIC50: 1.54E+4nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using linoleic acid as substrate by spectrophotometric assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584663(CHEMBL5090671)
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using arachidonic acid as substrate by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584666(CHEMBL5070865)
Affinity DataIC50: 2.33E+4nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using arachidonic acid as substrate by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584661(CHEMBL5087097)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using linoleic acid as substrate by spectrophotometric assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584665(CHEMBL5086474)
Affinity DataIC50: 4.33E+4nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using arachidonic acid as substrate by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584664(CHEMBL5070746)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using arachidonic acid as substrate by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584662(CHEMBL5088464)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using arachidonic acid as substrate by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584661(CHEMBL5087097)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli using arachidonic acid as substrate by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584668(CHEMBL5089414)
Affinity DataKi:  22nMAssay Description:Non-competitive inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli assessed as inhibition constant using linol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584663(CHEMBL5090671)
Affinity DataKi:  290nMAssay Description:Non-competitive inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli assessed as inhibition constant using linol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584667(CHEMBL5080282)
Affinity DataKi:  790nMAssay Description:Non-competitive inhibition of wild type rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli assessed as inhibition constant using linol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584667(CHEMBL5080282)
Affinity DataKi:  790nMAssay Description:Mixed mode inhibition of wild type Rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli assessed as inhibition constant using linoleic a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Rabbit)
Mirea Russian Technological University

Curated by ChEMBL
LigandPNGBDBM50584667(CHEMBL5080282)
Affinity DataKi:  3.13E+3nMAssay Description:Mixed mode inhibition of wild type Rabbit N-terminal His-tagged ALOX15 expressed in Escherichia coli assessed as inhibition constant using arachidoni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed