Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50017641
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM259897(US9505780, JQ-1)
Affinity DataIC50: 92nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603594(CHEMBL5205457)
Affinity DataIC50: 107nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603592(CHEMBL5170506)
Affinity DataIC50: 347nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603591(CHEMBL5190640)
Affinity DataIC50: 417nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603598(CHEMBL5178583)
Affinity DataIC50: 419nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603589(CHEMBL5203606)
Affinity DataIC50: 471nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603586(CHEMBL5186976)
Affinity DataIC50: 481nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603594(CHEMBL5205457)
Affinity DataIC50: 502nMAssay Description:Inhibition of His-tagged recombinant BRD3 (unknown origin) (11 to 166 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as substrate me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603593(CHEMBL5203164)
Affinity DataIC50: 504nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603597(CHEMBL5204216)
Affinity DataIC50: 514nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603590(CHEMBL5189496)
Affinity DataIC50: 559nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603588(CHEMBL5180321)
Affinity DataIC50: 578nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603587(CHEMBL5193638)
Affinity DataIC50: 674nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603594(CHEMBL5205457)
Affinity DataIC50: 718nMAssay Description:Inhibition of His-tagged recombinant BRD2 (unknown origin) (11 to 162 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as substrate me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603594(CHEMBL5205457)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of His-tagged recombinant BRDT (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as substrate me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain and PHD finger-containing protein 3(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603594(CHEMBL5205457)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of His-tagged recombinant BRPF3 (unknown origin) (11 to 188 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as substrate m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 1(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603594(CHEMBL5205457)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of His-tagged recombinant BRD1 (unknown origin) (11 to 190 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as substrate me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603578(CHEMBL5184904)
Affinity DataIC50: 2.44E+3nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603580(CHEMBL5172772)
Affinity DataIC50: 2.65E+3nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603585(CHEMBL5192176)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603595(CHEMBL5191169)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603596(CHEMBL5180717)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603584(CHEMBL5204547)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603583(CHEMBL5192506)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603582(CHEMBL5187128)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603581(CHEMBL5170192)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603579(CHEMBL5169983)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
West China Hospital of Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603577(CHEMBL5181084)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed