Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50016256
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM109086(US8604016, 670 | US9938267, Cmpd ID 670 | US107935...)
Affinity DataIC50: 310nMAssay Description:Inhibition of GLS-1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM50593582(CHEMBL5179292)
Affinity DataEC50:  3.96E+3nMAssay Description:Inhibition of human recombinant GLS-1 by measuring glutamate production incubated for 1 hr by fluorescence based multimode plate reader methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlutaminase liver isoform, mitochondrial(Human)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM50593582(CHEMBL5179292)
Affinity DataEC50:  1.29E+4nMAssay Description:Inhibition of human recombinant GLS-2 by measuring glutamate production incubated for 1 hr by fluorescence based multimode plate reader methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed