Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50016717
TargetAmine oxidase [flavin-containing] B(Human)
Swedish Defence Research Agency

Curated by ChEMBL
LigandPNGBDBM50093227(CHEMBL3586608)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human MAO-B expressed in Pichia pastoris using kynuramine as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Swedish Defence Research Agency

Curated by ChEMBL
LigandPNGBDBM50532731(CHEMBL4571763)
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant human MAO-B expressed in Pichia pastoris using kynuramine as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Swedish Defence Research Agency

Curated by ChEMBL
LigandPNGBDBM50532731(CHEMBL4571763)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human MAO-B expressed in Pichia pastoris using kynuramine as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Swedish Defence Research Agency

Curated by ChEMBL
LigandPNGBDBM50532731(CHEMBL4571763)
Affinity DataKi:  93nMAssay Description:Binding affinity to recombinant human MAO-B expressed in Pichia pastoris assessed as inhibition constant using benzylamine as substrate by Michaelis-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Swedish Defence Research Agency

Curated by ChEMBL
LigandPNGBDBM50093227(CHEMBL3586608)
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant human AChE by spectrophotometric Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Swedish Defence Research Agency

Curated by ChEMBL
LigandPNGBDBM50532731(CHEMBL4571763)
Affinity DataKi:  130nMAssay Description:Binding affinity to recombinant human MAO-B expressed in Pichia pastoris assessed as inhibition constant using benzylamine as substrate by Michaelis-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Swedish Defence Research Agency

Curated by ChEMBL
LigandPNGBDBM50532731(CHEMBL4571763)
Affinity DataKi:  190nMAssay Description:Binding affinity to recombinant human MAO-B expressed in Pichia pastoris assessed as inhibition constant using benzylamine as substrate by Michaelis-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Swedish Defence Research Agency

Curated by ChEMBL
LigandPNGBDBM50532731(CHEMBL4571763)
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant human MAO-B expressed in Pichia pastoris using kynuramine as substrate by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Mouse)
Swedish Defence Research Agency

Curated by ChEMBL
LigandPNGBDBM50093227(CHEMBL3586608)
Affinity DataIC50: 400nMAssay Description:Inhibition of recombinant mouse AChE expressed in human HEK293F cells using acetylthiocholine iodide as substrate by spectrophotometric Ellman's meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Mouse)
Swedish Defence Research Agency

Curated by ChEMBL
LigandPNGBDBM50532731(CHEMBL4571763)
Affinity DataIC50: 700nMAssay Description:Inhibition of recombinant mouse AChE expressed in human HEK293F cells using acetylthiocholine iodide as substrate by spectrophotometric Ellman's meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Swedish Defence Research Agency

Curated by ChEMBL
LigandPNGBDBM50532731(CHEMBL4571763)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of recombinant human AChE by spectrophotometric Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Swedish Defence Research Agency

Curated by ChEMBL
LigandPNGBDBM50532731(CHEMBL4571763)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of recombinant human AChE by spectrophotometric Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Mouse)
Swedish Defence Research Agency

Curated by ChEMBL
LigandPNGBDBM50532731(CHEMBL4571763)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant mouse AChE expressed in human HEK293F cells using acetylthiocholine iodide as substrate by spectrophotometric Ellman's meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Swedish Defence Research Agency

Curated by ChEMBL
LigandPNGBDBM50532731(CHEMBL4571763)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant human AChE by spectrophotometric Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Swedish Defence Research Agency

Curated by ChEMBL
LigandPNGBDBM50093227(CHEMBL3586608)
Affinity DataKi:  4.50E+3nMAssay Description:Tight binding inhibition of recombinant human MAO-B expressed in Pichia pastoris assessed as inhibition constant using benzylamine as substrate at 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed