Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50017727
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50371783(CHEMBL397237)
Affinity DataIC50: 13nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-binding incubated for 15 mins followed by addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604459(CHEMBL5195797)
Affinity DataIC50: 13nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-binding incubated for 15 mins followed by addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604458(CHEMBL5173775)
Affinity DataIC50: 44nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-binding incubated for 15 mins followed by addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50371783(CHEMBL397237)
Affinity DataIC50: 79nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-induced calcium response incubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604459(CHEMBL5195797)
Affinity DataIC50: 100nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-induced calcium response incubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604464(CHEMBL5183834)
Affinity DataIC50: 110nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-induced calcium response incubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604451(CHEMBL5186932)
Affinity DataIC50: 130nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-binding incubated for 15 mins followed by addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604453(CHEMBL5203743)
Affinity DataIC50: 250nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-binding incubated for 15 mins followed by addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604451(CHEMBL5186932)
Affinity DataIC50: 270nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-induced calcium response incubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604464(CHEMBL5183834)
Affinity DataIC50: 430nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-binding incubated for 15 mins followed by addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604458(CHEMBL5173775)
Affinity DataIC50: 660nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-induced calcium response incubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604454(CHEMBL5182926)
Affinity DataIC50: 1.06E+3nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-binding incubated for 15 mins followed by addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604453(CHEMBL5203743)
Affinity DataIC50: 2.49E+3nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-induced calcium response incubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604457(CHEMBL5179622)
Affinity DataIC50: 2.71E+3nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-binding incubated for 15 mins followed by addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604452(CHEMBL5171358)
Affinity DataIC50: 4.26E+3nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-binding incubated for 15 mins followed by addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604457(CHEMBL5179622)
Affinity DataIC50: 7.73E+3nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-induced calcium response incubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604454(CHEMBL5182926)
Affinity DataIC50: 1.57E+4nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-induced calcium response incubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604456(CHEMBL5179345)
Affinity DataIC50: 1.72E+4nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-binding incubated for 15 mins followed by addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604456(CHEMBL5179345)
Affinity DataIC50: 2.47E+4nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-induced calcium response incubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604452(CHEMBL5171358)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-induced calcium response incubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604465(CHEMBL5201451)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-binding incubated for 15 mins followed by addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604463(CHEMBL5174137)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-binding incubated for 15 mins followed by addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604455(CHEMBL5183117)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-induced calcium response incubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604462(CHEMBL5184465)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-binding incubated for 15 mins followed by addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604461(CHEMBL5203131)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-binding incubated for 15 mins followed by addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604460(CHEMBL5199496)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-binding incubated for 15 mins followed by addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604460(CHEMBL5199496)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-induced calcium response incubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604461(CHEMBL5203131)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-induced calcium response incubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604462(CHEMBL5184465)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-induced calcium response incubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604463(CHEMBL5174137)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-induced calcium response incubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604455(CHEMBL5183117)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-binding incubated for 15 mins followed by addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50604465(CHEMBL5201451)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to human CXCR2 expressed in human U87 cells assessed as inhibition of CXCL8 AF647-induced calcium response incubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed