Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50017223
TargetCytochrome P450 2C9(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50600340(CHEMBL5202937)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetCytochrome P450 3A4(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50600340(CHEMBL5202937)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin) using testosterone as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetCytochrome P450 1A2(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50600340(CHEMBL5202937)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetCytochrome P450 2C19(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50600340(CHEMBL5202937)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetCytochrome P450 2D6(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50600340(CHEMBL5202937)
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed