Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50016267
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50155926(CHEMBL3183703)
Affinity DataIC50: 13nMAssay Description:Inhibition of NLRP3 inflammasome activation in PMA differentiated LPS-primed human THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50593673(CHEMBL5207889)
Affinity DataIC50: 49nMAssay Description:Inhibition of NLRP3 inflammasome activation in PMA differentiated LPS-primed human THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50593663(CHEMBL5184033)
Affinity DataIC50: 60nMAssay Description:Inhibition of NLRP3 inflammasome activation in PMA differentiated LPS-primed human THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50593671(CHEMBL5188490)
Affinity DataIC50: 61nMAssay Description:Inhibition of NLRP3 inflammasome activation in PMA differentiated LPS-primed human THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50593674(CHEMBL5187589)
Affinity DataIC50: 100nMAssay Description:Inhibition of NLRP3 inflammasome activation in PMA differentiated LPS-primed human THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50593665(CHEMBL5184563)
Affinity DataIC50: 108nMAssay Description:Inhibition of NLRP3 inflammasome activation in PMA differentiated LPS-primed human THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50593662(CHEMBL5184899)
Affinity DataIC50: 146nMAssay Description:Inhibition of NLRP3 inflammasome activation in PMA differentiated LPS-primed human THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50593667(CHEMBL5188246)
Affinity DataIC50: 243nMAssay Description:Inhibition of NLRP3 inflammasome activation in PMA differentiated LPS-primed human THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50593668(CHEMBL5183540)
Affinity DataIC50: 247nMAssay Description:Inhibition of NLRP3 inflammasome activation in PMA differentiated LPS-primed human THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50593670(CHEMBL5207305)
Affinity DataIC50: 636nMAssay Description:Inhibition of NLRP3 inflammasome activation in PMA differentiated LPS-primed human THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50593666(CHEMBL5189690)
Affinity DataIC50: 641nMAssay Description:Inhibition of NLRP3 inflammasome activation in PMA differentiated LPS-primed human THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50593664(CHEMBL5179909)
Affinity DataIC50: 947nMAssay Description:Inhibition of NLRP3 inflammasome activation in PMA differentiated LPS-primed human THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50593669(CHEMBL5170114)
Affinity DataIC50: 2.38E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in PMA differentiated LPS-primed human THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50593672(CHEMBL5207084)
Affinity DataIC50: 9.18E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in PMA differentiated LPS-primed human THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed