Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50016487
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595298(CHEMBL5207902)
Affinity DataIC50: 540nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595300(CHEMBL5201191)
Affinity DataIC50: 570nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595297(CHEMBL5190035)
Affinity DataIC50: 670nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595301(CHEMBL5169865)
Affinity DataIC50: 820nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595310(CHEMBL5203265)
Affinity DataIC50: 920nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595311(CHEMBL5209321)
Affinity DataIC50: 960nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595319(CHEMBL5186222)
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595299(CHEMBL5201859)
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595312(CHEMBL5173485)
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595315(CHEMBL5183590)
Affinity DataIC50: 1.82E+3nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595298(CHEMBL5207902)
Affinity DataIC50: 2.06E+3nMAssay Description:Inhibition of human TRPC4 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595309(CHEMBL5192702)
Affinity DataIC50: 2.21E+3nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595330(CHEMBL5187515)
Affinity DataIC50: 2.21E+3nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595313(CHEMBL5171565)
Affinity DataIC50: 2.24E+3nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595316(CHEMBL5194092)
Affinity DataIC50: 2.27E+3nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595308(CHEMBL5206434)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595317(CHEMBL5202944)
Affinity DataIC50: 2.41E+3nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595320(CHEMBL5182312)
Affinity DataIC50: 2.64E+3nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595329(CHEMBL5194160)
Affinity DataIC50: 2.93E+3nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595321(CHEMBL5202586)
Affinity DataIC50: 2.95E+3nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595318(CHEMBL5176140)
Affinity DataIC50: 3.13E+3nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595322(CHEMBL5185813)
Affinity DataIC50: 3.35E+3nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595307(CHEMBL5191462)
Affinity DataIC50: 4.63E+3nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595324(CHEMBL5170000)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595331(CHEMBL5186146)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595305(CHEMBL5208734)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595328(CHEMBL5173272)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595327(CHEMBL5185490)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595326(CHEMBL5191534)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595325(CHEMBL5172936)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595314(CHEMBL5182054)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595323(CHEMBL5195015)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595306(CHEMBL5200070)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595302(CHEMBL5206422)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595304(CHEMBL5200061)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595303(CHEMBL5169949)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM49021(N-(furan-2-ylmethyl)-1-(phenylmethyl)benzimidazol-...)
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibition of human TRPC5 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM49021(N-(furan-2-ylmethyl)-1-(phenylmethyl)benzimidazol-...)
Affinity DataIC50: 7.72E+4nMAssay Description:Inhibition of human TRPC4 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed