Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50016775
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597108(CHEMBL5184251 | US20230287003, Example 1v)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597108(CHEMBL5184251 | US20230287003, Example 1v)
Affinity DataIC50: 12nMAssay Description:Inhibition of human C-terminal nanoLuc-tagged BCL6 expressed in HEK293T cells co-expressing HaloTagged-SMRT using NanoBRET furimazine as substrate in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM522280(US11161839, Example 10a)
Affinity DataIC50: 26nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597098(CHEMBL5173162 | US20230287003, Example 6b)
Affinity DataIC50: 39nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597100(CHEMBL5203649)
Affinity DataIC50: 78nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597103(CHEMBL5199127 | US20230287003, Example 6a)
Affinity DataIC50: 94nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597102(CHEMBL5178675 | US20230287003, Example 1a)
Affinity DataIC50: 130nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597098(CHEMBL5173162 | US20230287003, Example 6b)
Affinity DataIC50: 210nMAssay Description:Inhibition of human C-terminal nanoLuc-tagged BCL6 expressed in HEK293T cells co-expressing HaloTagged-SMRT using NanoBRET furimazine as substrate in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597105(CHEMBL5187360 | US20230287003, Example 1j)
Affinity DataIC50: 480nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597111(CHEMBL5171937)
Affinity DataIC50: 490nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM522280(US11161839, Example 10a)
Affinity DataIC50: 570nMAssay Description:Inhibition of human C-terminal nanoLuc-tagged BCL6 expressed in HEK293T cells co-expressing HaloTagged-SMRT using NanoBRET furimazine as substrate in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597099(CHEMBL5201812)
Affinity DataIC50: 610nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597100(CHEMBL5203649)
Affinity DataIC50: 670nMAssay Description:Inhibition of human C-terminal nanoLuc-tagged BCL6 expressed in HEK293T cells co-expressing HaloTagged-SMRT using NanoBRET furimazine as substrate in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597106(CHEMBL5186909)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597101(CHEMBL5207801 | US20230287003, Example 1b)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597104(CHEMBL5173975 | US20230287003, Example 1e)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50587558(CHEMBL5079963)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597118(CHEMBL5187292)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597107(CHEMBL5182117)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597113(CHEMBL5177733)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597102(CHEMBL5178675 | US20230287003, Example 1a)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human C-terminal nanoLuc-tagged BCL6 expressed in HEK293T cells co-expressing HaloTagged-SMRT using NanoBRET furimazine as substrate in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597119(CHEMBL5179621)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597117(CHEMBL5183596 | US20230287003, Example 9a)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597105(CHEMBL5187360 | US20230287003, Example 1j)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human C-terminal nanoLuc-tagged BCL6 expressed in HEK293T cells co-expressing HaloTagged-SMRT using NanoBRET furimazine as substrate in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597114(CHEMBL5185841)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597104(CHEMBL5173975 | US20230287003, Example 1e)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of human C-terminal nanoLuc-tagged BCL6 expressed in HEK293T cells co-expressing HaloTagged-SMRT using NanoBRET furimazine as substrate in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597115(CHEMBL5182834)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597101(CHEMBL5207801 | US20230287003, Example 1b)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of human C-terminal nanoLuc-tagged BCL6 expressed in HEK293T cells co-expressing HaloTagged-SMRT using NanoBRET furimazine as substrate in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597109(CHEMBL5198634)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597099(CHEMBL5201812)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of human C-terminal nanoLuc-tagged BCL6 expressed in HEK293T cells co-expressing HaloTagged-SMRT using NanoBRET furimazine as substrate in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597110(CHEMBL5197204)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597106(CHEMBL5186909)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of human C-terminal nanoLuc-tagged BCL6 expressed in HEK293T cells co-expressing HaloTagged-SMRT using NanoBRET furimazine as substrate in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597107(CHEMBL5182117)
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of human C-terminal nanoLuc-tagged BCL6 expressed in HEK293T cells co-expressing HaloTagged-SMRT using NanoBRET furimazine as substrate in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597103(CHEMBL5199127 | US20230287003, Example 6a)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human C-terminal nanoLuc-tagged BCL6 expressed in HEK293T cells co-expressing HaloTagged-SMRT using NanoBRET furimazine as substrate in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597112(CHEMBL5186317)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetB-cell lymphoma 6 protein(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50597116(CHEMBL5198681)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of human N-terminal thioredoxin 6-His tagged BCL6 BTB domain (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed