Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50017940
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606364(CHEMBL5185586)
Affinity DataKd:  210nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50571811(CHEMBL4856564)
Affinity DataKd:  230nMAssay Description:Binding affinity to recombinant N-terminal His6-tagged human KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli BL21 (DE3) by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50571811(CHEMBL4856564)
Affinity DataKd:  230nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606358(CHEMBL5184256)
Affinity DataKd:  480nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606368(CHEMBL5194748)
Affinity DataKd:  580nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606365(CHEMBL5206662)
Affinity DataKd:  710nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606362(CHEMBL5186985)
Affinity DataKd:  1.03E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606367(CHEMBL5208642)
Affinity DataKd:  1.08E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606357(CHEMBL5181879)
Affinity DataKd:  1.35E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606360(CHEMBL5184121)
Affinity DataKd:  1.42E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606359(CHEMBL5202487)
Affinity DataKd:  1.45E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606369(CHEMBL5170702)
Affinity DataKd:  1.48E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606350(CHEMBL5184030)
Affinity DataKd:  1.76E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606361(CHEMBL5209312)
Affinity DataKd:  2.08E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606351(CHEMBL5195730)
Affinity DataKd:  2.81E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606363(CHEMBL5185737)
Affinity DataKd:  2.91E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606366(CHEMBL5180035)
Affinity DataKd:  2.92E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606355(CHEMBL5201699)
Affinity DataKd:  6.11E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606354(CHEMBL5184384)
Affinity DataKd:  6.64E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606356(CHEMBL5200998)
Affinity DataKd:  8.94E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606353(CHEMBL5203318)
Affinity DataKd: >1.00E+4nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50606352(CHEMBL5207103)
Affinity DataKd: >1.00E+4nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Keap1-Nrf2 (322 to 609 residues) (unknown origin) protein-protein interaction expressed in Esc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed