Compile Data Set for Download or QSAR
Report error Found 85 Enz. Inhib. hit(s) with all data for entry = 50018680
TargetFree fatty acid receptor 3(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611320(CHEMBL5277000)
Affinity DataEC50:  220nMAssay Description:Agonist activity at FFA3 (unknown origin) expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetFree fatty acid receptor 2(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611316(CHEMBL5270112)
Affinity DataEC50:  740nMAssay Description:Agonist activity at FFA2 (unknown origin) expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetFree fatty acid receptor 2(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611317(CHEMBL5275861)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at FFA2 (unknown origin) expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetFree fatty acid receptor 2(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611318(CHEMBL5284951)
Affinity DataEC50:  380nMAssay Description:Agonist activity at FFA2 (unknown origin) expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetFree fatty acid receptor 3(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611316(CHEMBL5270112)
Affinity DataEC50:  220nMAssay Description:Agonist activity at FFA3 (unknown origin) expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetFree fatty acid receptor 3(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611317(CHEMBL5275861)
Affinity DataEC50:  220nMAssay Description:Agonist activity at FFA3 (unknown origin) expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetFree fatty acid receptor 3(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611318(CHEMBL5284951)
Affinity DataEC50:  220nMAssay Description:Agonist activity at FFA3 (unknown origin) expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetFree fatty acid receptor 3(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611319(CHEMBL5281556)
Affinity DataEC50:  220nMAssay Description:Agonist activity at FFA3 (unknown origin) expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetFree fatty acid receptor 3(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50337031(5-ethyl-2-mercapto-3H-pyrano[2,3-d]pyrimidine-4,7-...)
Affinity DataEC50:  220nMAssay Description:Agonist activity at FFA3 (unknown origin) expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetFree fatty acid receptor 3(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50384616(CHEMBL2036813)
Affinity DataEC50:  220nMAssay Description:Agonist activity at FFA3 (unknown origin) expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611316(CHEMBL5270112)
Affinity DataEC50:  51nMAssay Description:Agonist activity at human HCA2 expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611317(CHEMBL5275861)
Affinity DataEC50:  51nMAssay Description:Agonist activity at human HCA2 expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611318(CHEMBL5284951)
Affinity DataEC50:  51nMAssay Description:Agonist activity at human HCA2 expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611319(CHEMBL5281556)
Affinity DataEC50:  51nMAssay Description:Agonist activity at human HCA2 expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50337031(5-ethyl-2-mercapto-3H-pyrano[2,3-d]pyrimidine-4,7-...)
Affinity DataEC50:  51nMAssay Description:Agonist activity at human HCA2 expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611320(CHEMBL5277000)
Affinity DataEC50:  51nMAssay Description:Agonist activity at human HCA2 expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50384616(CHEMBL2036813)
Affinity DataEC50:  51nMAssay Description:Agonist activity at human HCA2 expressed in human Flp-In-293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50226181(Carbamic acid 5-hydroxy-6-{4-hydroxy-3-[4-hydroxy-...)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of Escherichia coli DNA gyraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611301(CHEMBL5287867)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of Escherichia coli DNA gyraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetAlbumin(Bovine)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611309(CHEMBL5278862)
Affinity DataIC50: 5.90nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetAlbumin(Bovine)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611303(CHEMBL5279919)
Affinity DataIC50: 8.90nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetAlbumin(Bovine)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611306(CHEMBL5271257)
Affinity DataIC50: 9.20nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetAlbumin(Bovine)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611307(CHEMBL5285447)
Affinity DataIC50: 9.30nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetAlbumin(Bovine)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611305(CHEMBL5272468)
Affinity DataIC50: 9.40nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetAlbumin(Bovine)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611310(CHEMBL5270068)
Affinity DataIC50: 11nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetAlbumin(Bovine)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611304(CHEMBL5266358)
Affinity DataIC50: 12nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetAlbumin(Bovine)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611311(CHEMBL5272008)
Affinity DataIC50: 12nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetAlbumin(Bovine)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611308(CHEMBL5290916)
Affinity DataIC50: 12nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetAlbumin(Bovine)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611302(CHEMBL5266328)
Affinity DataIC50: 13nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetAlbumin(Bovine)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50174201(ARTHROTEC | GP 45840 | SOLARAZE | Sodium; [2-(2,6-...)
Affinity DataIC50: 19nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611335(CHEMBL5279318)
Affinity DataIC50: 40nMAssay Description:Inhibition of sheep COX-2 by Cayman colorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 40nMAssay Description:Inhibition of sheep COX-2 by Cayman colorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611336(CHEMBL5274256)
Affinity DataIC50: 40nMAssay Description:Inhibition of sheep COX-2 by Cayman colorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611331(CHEMBL5271017)
Affinity DataIC50: 752nMAssay Description:Inhibition of DNA topoisomerase 2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611333(CHEMBL5275333)
Affinity DataIC50: 776nMAssay Description:Inhibition of DNA topoisomerase 2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611332(CHEMBL5282398)
Affinity DataIC50: 791nMAssay Description:Inhibition of DNA topoisomerase 2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM22984(Adriamycin | (8S,10S)-10-{[(2R,4S,5S,6S)-4-amino-5...)
Affinity DataIC50: 940nMAssay Description:Inhibition of DNA topoisomerase 2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611335(CHEMBL5279318)
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of 5-LOX (unknown origin) by colorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611336(CHEMBL5274256)
Affinity DataIC50: 1.93E+3nMAssay Description:Inhibition of 5-LOX (unknown origin) by colorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 3.34E+3nMAssay Description:Inhibition of 5-LOX (unknown origin) by colorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611323(CHEMBL5283904)
Affinity DataIC50: 3.61E+3nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hrs by colorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611327(CHEMBL5276959)
Affinity DataIC50: 3.61E+3nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hrs by colorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611322(CHEMBL5274535)
Affinity DataIC50: 4.06E+3nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hrs by colorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611334(CHEMBL5275837)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of recombinant human SIRT1 expressed in Escherichia coli using Fluor de Lys-SIRT1/2 substrate in presence of NAD+ by fluorescence micropla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50309832(2H-chromeno[2,3-d]pyrimidine-2,4(3H)-dione | CHEMB...)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of recombinant human SIRT1 expressed in Escherichia coli using Fluor de Lys-SIRT1/2 substrate in presence of NAD+ by fluorescence micropla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)
Affinity DataIC50: 5.77E+3nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hrs by colorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50309831(10-Phenyl-7-oxa-8,10-diaza-benzo[a]anthracene-9,11...)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of recombinant human SIRT1 expressed in Escherichia coli using Fluor de Lys-SIRT1/2 substrate in presence of NAD+ by fluorescence micropla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611312(CHEMBL5291178)
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase assessed as decrease in release of p-nitrophenol using pNPG as substrate incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611325(CHEMBL5277605)
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hrs by colorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50611314(CHEMBL5278001)
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae alpha-glucosidase assessed as decrease in release of p-nitrophenol using pNPG as substrate incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
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