Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50017943
TargetSigma intracellular receptor 2(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50606398(Metarrestin | Ml-246 | ML-246)
Affinity DataKi:  244nMAssay Description:Binding affinity to sigma2 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetAlpha-2C adrenergic receptor(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50606398(Metarrestin | Ml-246 | ML-246)
Affinity DataKi:  1.22E+3nMAssay Description:Binding affinity to alpha2C receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50606398(Metarrestin | Ml-246 | ML-246)
Affinity DataKi:  3.26E+3nMAssay Description:Binding affinity to alpha1D receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50606398(Metarrestin | Ml-246 | ML-246)
Affinity DataKi:  3.41E+3nMAssay Description:Binding affinity to DAT receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetHistamine H1 receptor(Human)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50606398(Metarrestin | Ml-246 | ML-246)
Affinity DataKi:  3.56E+3nMAssay Description:Binding affinity to H1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed