Compile Data Set for Download or QSAR
Report error Found 61 Enz. Inhib. hit(s) with all data for entry = 50016809
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597385(CHEMBL5169323)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597397(CHEMBL5194755)
Affinity DataKi:  13nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597392(CHEMBL5208709)
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597391(CHEMBL5186338)
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597385(CHEMBL5169323)
Affinity DataKi:  14nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597390(CHEMBL5204680)
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597388(CHEMBL5177782)
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597394(CHEMBL5178465)
Affinity DataKi:  21nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597393(CHEMBL5184362)
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597384(CHEMBL5191017)
Affinity DataKi:  21nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597386(CHEMBL5207081)
Affinity DataKi:  33nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM512835(acs.jmedchem.1c00409_ST.430)
Affinity DataIC50: 34nMAssay Description:Inhibition of his-tagged SARS CoV-2 main protease expressed in HEK cells using Boc-Abu-Tle-Leu-Gln-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597382(CHEMBL5207392)
Affinity DataKi:  34nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597381(CHEMBL4855437)
Affinity DataIC50: 34nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597379(CHEMBL5189863)
Affinity DataKi:  36nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597399(CHEMBL5178568)
Affinity DataKi:  42nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597375(CHEMBL5204452)
Affinity DataKi:  43nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597400(CHEMBL5197891)
Affinity DataKi:  51nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597372(CHEMBL5188939)
Affinity DataIC50: 55nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597370(CHEMBL5189565)
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597371(CHEMBL5173920)
Affinity DataIC50: 72nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597395(CHEMBL5192654)
Affinity DataKi:  73nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597368(CHEMBL5204130)
Affinity DataKi:  74nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597378(CHEMBL5202104)
Affinity DataKi:  77nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597376(CHEMBL5204064)
Affinity DataKi:  84nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597386(CHEMBL5207081)
Affinity DataIC50: 88nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597400(CHEMBL5197891)
Affinity DataIC50: 89nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597375(CHEMBL5204452)
Affinity DataIC50: 91nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597395(CHEMBL5192654)
Affinity DataIC50: 117nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597377(CHEMBL5207613)
Affinity DataKi:  119nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597399(CHEMBL5178568)
Affinity DataIC50: 125nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597368(CHEMBL5204130)
Affinity DataIC50: 143nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597376(CHEMBL5204064)
Affinity DataIC50: 147nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597373(CHEMBL5199191)
Affinity DataIC50: 159nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597398(CHEMBL5181137)
Affinity DataKi:  161nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597396(CHEMBL5186708)
Affinity DataIC50: 166nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597372(CHEMBL5188939)
Affinity DataKi:  186nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597398(CHEMBL5181137)
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597383(CHEMBL5192027)
Affinity DataIC50: 235nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597373(CHEMBL5199191)
Affinity DataKi:  250nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597382(CHEMBL5207392)
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597397(CHEMBL5194755)
Affinity DataIC50: 255nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597378(CHEMBL5202104)
Affinity DataIC50: 281nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597389(CHEMBL5169680)
Affinity DataIC50: 288nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597374(CHEMBL5199531)
Affinity DataKi:  295nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM429304(jm5b01461, Compound 124 | indole chloropyridinyl-e...)
Affinity DataIC50: 313nMAssay Description:Inhibition of his-tagged SARS CoV-2 main protease expressed in HEK cells using Boc-Abu-Tle-Leu-Gln-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597379(CHEMBL5189863)
Affinity DataIC50: 316nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597374(CHEMBL5199531)
Affinity DataIC50: 349nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597371(CHEMBL5173920)
Affinity DataKi:  393nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 assessed as inhibition constant using Boc-Abu-Tle-Le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50597384(CHEMBL5191017)
Affinity DataIC50: 454nMAssay Description:Inhibition of recombinant his tagged SARS CoV-2 main protease expressed in Escherichia coli BL21 using Boc-Abu-Tle-Leu-Gln-AMC37 as fluorogenic subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
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