Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50016122
TargetSerine/threonine-protein kinase pim-1(Human)
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of Pim-1 (unknown origin) measured by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of Pim-1 (unknown origin) measured by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Inhibition of Pim-1 (unknown origin) measured by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of Pim-1 (unknown origin) measured by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 176nMAssay Description:Inhibition of Pim-1 (unknown origin) measured by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of Pim-1 (unknown origin) measured by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 434nMAssay Description:Inhibition of Pim-1 (unknown origin) measured by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 468nMAssay Description:Inhibition of Pim-1 (unknown origin) measured by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 881nMAssay Description:Inhibition of Pim-1 (unknown origin) measured by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 2.19E+3nMAssay Description:Inhibition of Pim-1 (unknown origin) measured by ADP-Glo kinase assayMore data for this Ligand-Target Pair



3D Structure (crystal)





