Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50017431
TargetProlyl endopeptidase FAP(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50326390((2S,4S)-1-({(2S,4S)-4-[2-(1,3-Dihydro-2H-isoindol-...)
Affinity DataIC50: 20nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataIC50: 22nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProlyl endopeptidase FAP(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50431242(CHEMBL2333026)
Affinity DataIC50: 36nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50155838((S)-1-((S)-1-(4-phenylbutanoyl)pyrrolidine-2-carbo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProlyl endopeptidase FAP(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50155838((S)-1-((S)-1-(4-phenylbutanoyl)pyrrolidine-2-carbo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM11695((2S)-1-{2-[(3-hydroxyadamantan-1-yl)amino]acetyl}p...)
Affinity DataIC50: 120nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50326390((2S,4S)-1-({(2S,4S)-4-[2-(1,3-Dihydro-2H-isoindol-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProlyl endopeptidase FAP(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM11695((2S)-1-{2-[(3-hydroxyadamantan-1-yl)amino]acetyl}p...)
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProlyl endopeptidase FAP(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50431227(CHEMBL2333024)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProlyl endopeptidase FAP(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50200721((R)-1-(2-(cyclohexanecarboxamido)acetyl)pyrrolidin...)
Affinity DataKi:  14nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProlyl endopeptidase FAP(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataKi:  66nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProlyl endopeptidase FAP(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50382283(CHEMBL2022530 | US9346814, Ref. Cmpd No 1 (Example...)
Affinity DataKi:  110nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProlyl endopeptidase FAP(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50601877(CHEMBL5171879)
Affinity DataKi:  200nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProlyl endopeptidase FAP(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50601879(CHEMBL5199424)
Affinity DataKi:  720nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProlyl endopeptidase FAP(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50601876(CHEMBL5195493)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50200721((R)-1-(2-(cyclohexanecarboxamido)acetyl)pyrrolidin...)
Affinity DataKi:  9.08E+3nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProlyl endopeptidase FAP(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50601875(CHEMBL5172375)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProlyl endopeptidase FAP(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50601878(CHEMBL5192850)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProlyl endopeptidase FAP(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50601874(CHEMBL5175365)
Affinity DataKi: >2.50E+4nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50382283(CHEMBL2022530 | US9346814, Ref. Cmpd No 1 (Example...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed