Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50015799
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50357312(IBRUTINIB | US9181263, 1 | US9108973, Ref 1 | US92...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589601(CHEMBL5180302)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589602(CHEMBL5192748)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589603(CHEMBL5195504)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589588(CHEMBL5208265)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589624(CHEMBL5193942)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589600(CHEMBL5206496)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589605(CHEMBL5204458)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589607(CHEMBL5170025)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589626(CHEMBL5177044)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589613(CHEMBL5196932)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589616(CHEMBL5176551)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589625(CHEMBL5198455)
Affinity DataIC50: 1nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589611(CHEMBL5170833)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589622(CHEMBL5189426)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589619(CHEMBL5189231)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589610(CHEMBL5196670)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589612(CHEMBL5178389)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589606(CHEMBL5193597)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589627(CHEMBL5202754)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589617(CHEMBL5179204)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589624(CHEMBL5193942)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of BTK in human TMD8 cells assessed as inhibition of BTK autophosphorylation at Tyr223 measured by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589604(CHEMBL5205889)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM291522(US9580449, Example A39 | 1-(4-(((6-amino-5-(4-phen...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589592(CHEMBL5206716)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589623(CHEMBL5179080)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589618(CHEMBL5193930)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589608(CHEMBL5175574)
Affinity DataIC50: 2nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589620(CHEMBL5187153)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589621(CHEMBL5206497)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589598(CHEMBL5206093)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589614(CHEMBL5188524)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589594(CHEMBL5171858)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589586(CHEMBL5203573)
Affinity DataIC50: 8.40nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589615(CHEMBL5179333)
Affinity DataIC50: 11nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589589(CHEMBL5208592)
Affinity DataIC50: 16nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589583(CHEMBL5179757)
Affinity DataIC50: 17nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589609(CHEMBL5184628)
Affinity DataIC50: 23nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589587(CHEMBL5183474)
Affinity DataIC50: 26nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM139991(US8901140, 5 | US9358227, 5)
Affinity DataIC50: 32nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589584(CHEMBL5191643)
Affinity DataIC50: 52nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589595(CHEMBL5206968)
Affinity DataIC50: 69nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589599(CHEMBL5197246)
Affinity DataIC50: 93nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM161389(US9108973, 2 | US10124003, Ref. Ex. Compound 3 | U...)
Affinity DataIC50: 95nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589585(CHEMBL5184198)
Affinity DataIC50: 99nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589593(CHEMBL5187334)
Affinity DataIC50: 153nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589590(CHEMBL5188432)
Affinity DataIC50: 593nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589591(CHEMBL5198805)
Affinity DataIC50: 974nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589624(CHEMBL5193942)
Affinity DataIC50: 4.38E+3nMAssay Description:Inhibition of hERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50589596(CHEMBL5191588)
Affinity DataIC50: 5.41E+3nMAssay Description:Inhibition of BTK (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
Displayed 1 to 50 (of 51 total ) | Next | Last >>
Jump to: