Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50017999
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Dr. Harisingh Gour University

Curated by ChEMBL
LigandPNGBDBM469269(US10807985, Compound 44 | US20250129067, Compound ...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of ABCG2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Dr. Harisingh Gour University

Curated by ChEMBL
LigandPNGBDBM50606901(CHEMBL3394488)
Affinity DataIC50: 41nMAssay Description:Inhibition of ABCG2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Dr. Harisingh Gour University

Curated by ChEMBL
LigandPNGBDBM50606903(CHEMBL5218863)
Affinity DataIC50: 62nMAssay Description:Inhibition of ABCG2 (unknown origin) overexpressing in dog MDCK-II-BCRP cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Dr. Harisingh Gour University

Curated by ChEMBL
LigandPNGBDBM50085526(4-[2-(3,5-dimethoxyphenyl)-(E)-1-ethenyl]-1,2-dime...)
Affinity DataIC50: 160nMAssay Description:Inhibition of wildtype ABCG2 (unknown origin) transfected in HEK293 cells measured after 30 mins by flow cytometric anlaysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Dr. Harisingh Gour University

Curated by ChEMBL
LigandPNGBDBM50595119(CHEMBL163972 | CHEBI:2161 | 6-Prenylchrysin)
Affinity DataIC50: 290nMAssay Description:Inhibition of ABCG2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Dr. Harisingh Gour University

Curated by ChEMBL
LigandPNGBDBM50606905(CHEMBL464796)
Affinity DataIC50: 2.97E+4nMAssay Description:Inhibition of ABCG2 (unknown origin) in Sf9 membrane vesicles using [3H] methotrexate as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Dr. Harisingh Gour University

Curated by ChEMBL
LigandPNGBDBM50606904(CHEMBL464795)
Affinity DataIC50: 4.17E+4nMAssay Description:Inhibition of ABCG2 (unknown origin) in Sf9 membrane vesicles using [3H] methotrexate as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Dr. Harisingh Gour University

Curated by ChEMBL
LigandPNGBDBM50606902(CHEMBL5219884)
Affinity DataIC50: 4.31E+4nMAssay Description:Inhibition of ABCG2 (unknown origin) overexpressing in dog MDCK-II-BCRP cells measured after 30 mins by flow cytometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed