Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50019488
TargetEndothelin-1 receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50122676(N-[2'-(4,5-Dimethyl-isoxazol-3-ylsulfamoyl)-4-oxaz...)
Affinity DataKi:  10nMAssay Description:Antagonist activity at human ETA receptor expressed in CHO cells assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetCholecystokinin(Rat)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50019777(7-(9-Hydroxy-2-isobutyl-3-oxo-2,3,9,9a-tetrahydro-...)
Affinity DataIC50: 1.40E+3nMAssay Description:Antagonist activity at 125I-labeled CCK-33 in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetCholecystokinin(Rat)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50014888(CHEMBL316561 | 4-Benzoylamino-4-dipropylcarbamoyl-...)
Affinity DataIC50: 6.00E+5nMAssay Description:Antagonist activity at 125I-labeled CCK-33 in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed