Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50020114
TargetTranscriptional coactivator YAP1(Homo sapiens)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of YAP (unknown origin) incubated for 24 hrs by Promega Dual-Luciferase Reporter AssayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of Avi-His-tagged human TEAD4 (217 to 434 residues)/N-biotinylated-N-terminal Cy5-labelled human YAP (60 to 100 residues) incubated for 1 ...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of Avi-His-tagged human TEAD4 (217 to 434 residues)/N-biotinylated-N-terminal Cy5-labelled human YAP (60 to 100 residues) incubated for 1 ...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of Avi-His-tagged human TEAD4 (217 to 434 residues)/N-biotinylated-N-terminal Cy5-labelled human YAP (60 to 100 residues) incubated for 1 ...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 6.20nMAssay Description:Binding affinity to SA sensor chip immobilized N-terminal avi-tagged biotinylated TEAD2 YAP binding domain (unknown origin) assessed as binding const...More data for this Ligand-Target Pair
TargetTranscriptional coactivator YAP1(Homo sapiens)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of YAP in HEK293T cells incubated for 24 hrs by Promega Dual-Luciferase Reporter AssayMore data for this Ligand-Target Pair
TargetTranscriptional coactivator YAP1(Homo sapiens)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of YAP in HEK293T cells incubated for 24 hrs by Promega Dual-Luciferase Reporter AssayMore data for this Ligand-Target Pair
TargetTranscriptional coactivator YAP1(Homo sapiens)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of YAP in HEK293T cells incubated for 24 hrs by Promega Dual-Luciferase Reporter AssayMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-1(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of His-tagged TEAD1 (unknown origin) preincubated for 30 mins followed by biotinylated lipid pocket addition and measured after 60 mins by...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of His-tagged TEAD2 (unknown origin) preincubated for 30 mins followed by biotinylated lipid pocket addition and measured after 60 mins by...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-1(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of His-tagged TEAD1 (unknown origin) preincubated for 30 mins followed by biotinylated lipid pocket addition and measured after 60 mins by...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-1(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of His-tagged TEAD1 (unknown origin) preincubated for 30 mins followed by biotinylated lipid pocket addition and measured after 60 mins by...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-5(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of His-tagged TEAD3 (unknown origin) preincubated for 30 mins followed by biotinylated lipid pocket addition and measured after 60 mins by...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-5(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of His-tagged TEAD3 (unknown origin) preincubated for 30 mins followed by biotinylated lipid pocket addition and measured after 60 mins by...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of His-tagged TEAD2 (unknown origin) preincubated for 30 mins followed by biotinylated lipid pocket addition and measured after 60 mins by...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of His-tagged TEAD2 (unknown origin) preincubated for 30 mins followed by biotinylated lipid pocket addition and measured after 60 mins by...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-3(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of His-tagged TEAD4 (unknown origin) preincubated for 30 mins followed by biotinylated lipid pocket addition and measured after 60 mins by...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-3(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of His-tagged TEAD4 (unknown origin) preincubated for 30 mins followed by biotinylated lipid pocket addition and measured after 60 mins by...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-5(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of His-tagged TEAD3 (unknown origin) preincubated for 30 mins followed by biotinylated lipid pocket addition and measured after 60 mins by...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-3(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of His-tagged TEAD4 (unknown origin) preincubated for 30 mins followed by biotinylated lipid pocket addition and measured after 60 mins by...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-1(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of TEAD1 mediating gene expression in human MCF7 cells incubated overnight by luciferase reporter assayMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-1(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of TEAD1 mediating gene expression in human MCF7 cells incubated overnight by luciferase reporter assayMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-1(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of TEAD1 mediating gene expression in human MCF7 cells incubated overnight by luciferase reporter assayMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-1(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of TEAD1 mediated gene transcription in human MCF7 cells incubated overnight by luciferase reporter assayMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-1(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of TEAD1 mediated gene transcription in human MCF7 cells incubated overnight by luciferase reporter assayMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-1(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of TEAD1 mediated gene transcription in human MCF7 cells incubated overnight by luciferase reporter assayMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-5(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of N-terminal 6xHis-tagged human TEAD3 auto palmitoylation (209 to 426 residues) expressed in Escherichia coli BL21 (DE3) cells by ABPP as...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 229nMAssay Description:Binding affinity to SA sensor chip immobilized N-terminal avi-tagged biotinylated TEAD2 YAP binding domain (unknown origin) assessed as binding const...More data for this Ligand-Target Pair
TargetTranscriptional coactivator YAP1(Homo sapiens)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 340nMAssay Description:Binding affinity to N-terminal YAP ( 1 to 291 residues) (unknown origin) expressed in Escherichia coli Rosetta cells assessed as dissociation constan...More data for this Ligand-Target Pair
TargetTranscriptional coactivator YAP1(Homo sapiens)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 391nMAssay Description:Inhibition of YAP (unknown origin) incubated for 24 hrs by Promega Dual-Luciferase Reporter AssayMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-3(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibition of N-terminal His-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-codonPlus (DE3)-RIPL cells by fluorescence p...More data for this Ligand-Target Pair
TargetTranscriptional coactivator YAP1(Homo sapiens)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 454nMAssay Description:Inhibition of YAP (unknown origin) incubated for 24 hrs by Promega Dual-Luciferase Reporter AssayMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-1(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Inhibition of N-terminal 6xHis-tagged human TEAD1 auto palmitoylation (209 to 426 residues) expressed in Escherichia coli BL21 (DE3) cells by ABPP as...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-5(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Inhibition of N-terminal 6xHis-tagged human TEAD3 auto palmitoylation (209 to 426 residues) expressed in Escherichia coli BL21 (DE3) cells by ABPP as...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 710nMAssay Description:Inhibition of TEAD2 (unknown origin) palmitoylation in the presence of alkyne-palmitoyl-CoAMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-5(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of N-terminal 6xHis-tagged human TEAD3 auto palmitoylation (209 to 426 residues) expressed in Escherichia coli BL21 (DE3) cells by ABPP as...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-3(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 2.60E+3nMAssay Description:Binding affinity to CM5 chip immobilised N-terminal histidine -tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli (DE3) cells ass...More data for this Ligand-Target Pair
TargetTranscriptional coactivator YAP1(Homo sapiens)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 2.64E+3nMAssay Description:Binding affinity to YAP WW domain (165 to 271 residues) (unknown origin) expressed in Escherichia coli Rosetta cells assessed as dissociation constan...More data for this Ligand-Target Pair
TargetTranscriptional coactivator YAP1(Homo sapiens)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of FAM-labelled GST-tagged full-length YAP (60 to 99 residues)(unknown origin)/N-terminal His-tagged TEAD2(217 to 447 residues) (unknown o...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of FAM-labelled GST-tagged full-length YAP (60 to 99 residues)(unknown origin)/GST-tagged TEAD4 (217 to 434 residues) (unknown origin) exp...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-1(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 9.40E+3nMAssay Description:Binding affinity to full-length His-tagged TEAD1 (unknown origin) assessed as dissociation constant by SPR assayMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-5(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 9.80E+3nMAssay Description:Binding affinity to TEAD 3 (unknown origin) assessed as dissociation constant by fluorescence polarisation assayMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-3(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 1.00E+4nMAssay Description:Binding affinity to CM5 chip immobilised N-terminal histidine -tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli (DE3) cells ass...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-5(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 1.60E+4nMAssay Description:Binding affinity to TEAD 3 (unknown origin) assessed as dissociation constant by fluorescence polarisation assayMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-3(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 2.80E+4nMAssay Description:Binding affinity to His-tagged TEAD4 YAP-binding domain (217 to 434 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by isot...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-3(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 2.94E+4nMAssay Description:Binding affinity to TEAD 4 (unknown origin) assessed as dissociation constant by fluorescence polarisation assayMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-3(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 3.10E+4nMAssay Description:Binding affinity to His-tagged TEAD4 YAP-binding domain (217 to 434 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by isot...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 3.50E+4nMAssay Description:Binding affinity to TEAD2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-3(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 3.70E+4nMAssay Description:Binding affinity to TEAD 4 (unknown origin) assessed as dissociation constant by fluorescence polarisation assayMore data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-3(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 7.30E+4nMAssay Description:Binding affinity to His-tagged TEAD4 YAP-binding domain (217 to 434 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by isot...More data for this Ligand-Target Pair





3D Structure (crystal)





























