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Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50015984
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM191600(US9714230, 89 | 2-(5-((4-chloro-2-methylbenzyl)oxy...)
Affinity DataIC50: 2nMAssay Description:Inhibition of full length human KDM5B expressed in baculovirus expression system using (ARTK(me3)QTARKSTGGKAPRKQLA peptide substMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455 | US20240139197, Compound 3)
Affinity DataIC50: 3nMAssay Description:Inhibition of full length human KDM5B expressed in baculovirus expression system using (ARTK(me3)QTARKSTGGKAPRKQLA peptide substMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590979(CHEMBL5206280)
Affinity DataIC50: 44nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590960(CHEMBL5182528)
Affinity DataIC50: 49nMAssay Description:Inhibition of recombinant KDM5B (residues 26 to 770) (unknown origin) transfected in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590961(CHEMBL5178382)
Affinity DataIC50: 52nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590980(CHEMBL5187685)
Affinity DataIC50: 52nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM281089(US10022354, Example 29)
Affinity DataIC50: 60nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590981(CHEMBL5180813)
Affinity DataIC50: 63nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590968(CHEMBL5174375)
Affinity DataIC50: 67nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590982(CHEMBL5190057)
Affinity DataIC50: 68nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5A(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590979(CHEMBL5206280)
Affinity DataIC50: 79nMAssay Description:Inhibition of KDM5A (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590963(CHEMBL5208852)
Affinity DataIC50: 89nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590970(CHEMBL5208099)
Affinity DataIC50: 105nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590965(CHEMBL5174240)
Affinity DataIC50: 109nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590978(CHEMBL5207005)
Affinity DataIC50: 114nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590984(CHEMBL5197642)
Affinity DataIC50: 139nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590962(CHEMBL5209413)
Affinity DataIC50: 146nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590971(CHEMBL5203703)
Affinity DataIC50: 166nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590967(CHEMBL5182152)
Affinity DataIC50: 209nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590964(CHEMBL5202845)
Affinity DataIC50: 219nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590972(CHEMBL5180165)
Affinity DataIC50: 243nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590986(CHEMBL5204336)
Affinity DataIC50: 330nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590969(CHEMBL5202556)
Affinity DataIC50: 346nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5C(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590979(CHEMBL5206280)
Affinity DataIC50: 353nMAssay Description:Inhibition of KDM5C (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590983(CHEMBL5195869)
Affinity DataIC50: 393nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590977(CHEMBL5192944)
Affinity DataIC50: 414nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590975(CHEMBL5193645)
Affinity DataIC50: 584nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590976(CHEMBL5183542)
Affinity DataIC50: 712nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590973(CHEMBL5200113)
Affinity DataIC50: 800nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590987(CHEMBL5200296)
Affinity DataIC50: 943nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590988(CHEMBL5208077)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590966(CHEMBL5209387)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590985(CHEMBL5175152)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50590974(CHEMBL5180353)
Affinity DataIC50: 4.43E+3nMAssay Description:Inhibition of KDM5B (unknown origin) incubated for 30 mins by HRTF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetLysine-specific demethylase 5B(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM26106(CHEMBL90852 | Oxalylglycine | [(carboxymethyl)carb...)
Affinity DataIC50: 2.45E+4nMAssay Description:Inhibition of KDM5B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMedPDB3D3D Structure (crystal)