Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50018007
TargetProtein kinase C delta type(Human)
Kagawa University

Curated by ChEMBL
LigandPNGBDBM50327944((1S,3R,5R,9R,13R)-9-Hydroxymethyl-16,16-dimethyl-3...)
Affinity DataKi:  9.80nMAssay Description:Inhibition of [3H]-PDBu binding to PKCdelta C1B domain (unknown origin) by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetProtein kinase C delta type(Human)
Kagawa University

Curated by ChEMBL
LigandPNGBDBM50606923(CHEMBL5220744)
Affinity DataKi:  17nMAssay Description:Inhibition of [3H]-PDBu binding to PKCdelta C1B domain (unknown origin) by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetProtein kinase C alpha type(Human)
Kagawa University

Curated by ChEMBL
LigandPNGBDBM50606923(CHEMBL5220744)
Affinity DataKi:  88nMAssay Description:Inhibition of [3H]-PDBu binding to PKCalpha C1A domain (unknown origin) by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetProtein kinase C alpha type(Human)
Kagawa University

Curated by ChEMBL
LigandPNGBDBM50606922(CHEMBL5219806)
Affinity DataKi:  100nMAssay Description:Inhibition of [3H]-PDBu binding to PKCalpha C1A domain (unknown origin) by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetProtein kinase C alpha type(Human)
Kagawa University

Curated by ChEMBL
LigandPNGBDBM50327944((1S,3R,5R,9R,13R)-9-Hydroxymethyl-16,16-dimethyl-3...)
Affinity DataKi:  120nMAssay Description:Inhibition of [3H]-PDBu binding to PKCalpha C1A domain (unknown origin) by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetProtein kinase C delta type(Human)
Kagawa University

Curated by ChEMBL
LigandPNGBDBM50606922(CHEMBL5219806)
Affinity DataKi:  130nMAssay Description:Inhibition of [3H]-PDBu binding to PKCdelta C1B domain (unknown origin) by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed