Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50019941
TargetMelatonin receptor type 1B(Human)
University of Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50343597(N-[2-(7-Pyridin-3-yl-1,6-dihydro-2H-indeno[5,4-b]f...)
Affinity DataKi:  0.0340nMAssay Description:Displacement of 2-[125I]iodoMLT from human MT2 receptor stably expressed in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50343597(N-[2-(7-Pyridin-3-yl-1,6-dihydro-2H-indeno[5,4-b]f...)
Affinity DataKi:  0.0690nMAssay Description:Displacement of 2-[125I]iodoMLT from human MT1 receptor stably expressed in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50624862(CHEMBL3103594)
Affinity DataKi:  0.210nMAssay Description:Binding affinity to MT2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50624862(CHEMBL3103594)
Affinity DataKi:  0.870nMAssay Description:Binding affinity to MT1 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50624861(CHEMBL5415352)
Affinity DataKi:  3.5nMAssay Description:Displacement of 2-[125I]iodoMLT from human MT2 receptor stably expressed in CHO cells incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50114726(N-[2-(5-Methoxy-2-pyridin-3-ylmethyl-benzofuran-3-...)
Affinity DataKi:  3.5nMAssay Description:Displacement of 2-[125I]iodoMLT from human MT2 receptor stably expressed in HEK cells incubated for 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50114726(N-[2-(5-Methoxy-2-pyridin-3-ylmethyl-benzofuran-3-...)
Affinity DataKi:  29nMAssay Description:Displacement of 2-[125I]iodoMLT from human MT1 receptor stably expressed in HEK cells incubated for 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50624861(CHEMBL5415352)
Affinity DataKi: >100nMAssay Description:Displacement of 2-[125I]iodoMLT from human MT1 receptor stably expressed in CHO cells incubated for 60 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed